SCHEMBL23771069

SCHEMBL23771069

O=C(Nc1ccc(Oc2ccnc3cc(OCCCC4=NC4)c4c(c23)OCCO4)cc1Cl)c1cccn(-c2ccc(F)cc2)c1=O

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.54
RET P07949 7/20 0.52
MET P08581 5/20 0.45
RIPK3 Q9Y572 4/20 0.45
RIPK1 Q13546 2/20 0.45
AURKA O14965 1/20 0.45
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
RIPK2 O43353 1/20 0.43
MST1R Q04912 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23749307 0.90 KDR (0.54) KDRRETMETRIPK3RIPK1
SCHEMBL23749275 0.90 KDR (0.53) KDRRETMETRIPK3RIPK1
SCHEMBL23749360 0.89 KDR (0.62) KDRRETMETRIPK3RIPK1
SCHEMBL23749435 0.89 KDR (0.69) KDRRETMETRIPK3RIPK1
SCHEMBL23771036 0.89 RET (0.55) KDRRETMETRIPK3RIPK1
SCHEMBL23749277 0.89 RET (0.58) KDRRETMETRIPK3RIPK1
SCHEMBL23749417 0.88 KDR (0.51) KDRRETMETRIPK3RIPK1
SCHEMBL23749362 0.83 RET (0.47) KDRRETMETRIPK3RIPK1
SCHEMBL23749289 0.81 MST1R (0.62) KDRRETMETMST1R
SCHEMBL23749440 0.79 RET (0.59) KDRRETMETMST1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3865487-A1 AROMATIC RING-LINKED DIOXANE-QUINAZOLINE OR -QUINOLINE COMPOUNDS, COMPOSITIONS AND USE THEREOF Beijing Scitech-MQ Pharmaceuticals Limited (CN) 2021-08-18 EP disclosed