SCHEMBL2379388

SCHEMBL2379388

CCOc1cc(C(=O)O)ccc1OCCCCOc1ccc2c(=O)n(C3CCCC3)sc2c1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MPI P34949 1/20 0.53
POLB P06746 1/20 0.49
CASP6 P55212 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
PDE4B Q07343 3/20 0.42
PDE4A P27815 2/20 0.42
PDE4C Q08493 2/20 0.42
PDE4D Q08499 2/20 0.42
DNMT3A Q9Y6K1 1/20 0.42
TSHR P16473 1/20 0.42
PPARD Q03181 1/20 0.39
PLA2G4B P0C869 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL787280 0.92 MPI (0.60) MPICYP1A2CYP2C9PDE4BPDE4A
SCHEMBL805880 0.88 MPI (0.60) MPICYP1A2CYP2C9PDE4BPDE4A
SCHEMBL787586 0.85 MPI (0.58) MPICYP1A2CYP2C9PDE4BPDE4A
SCHEMBL805879 0.84 CYP1A2 (0.58) MPIPOLBCYP1A2CYP2C9PLA2G4B
SCHEMBL804299 0.80 MPI (0.67) MPICYP1A2CYP2C9PDE4BPDE4A
SCHEMBL804302 0.80 MPI (0.65) MPICYP1A2CYP2C9DNMT3A
SCHEMBL787404 0.75 CYP1A2 (0.65) MPICYP1A2CYP2C9
SCHEMBL804282 0.74 CYP1A2 (0.77) MPICYP1A2CYP2C9
SCHEMBL787090 0.73 CYP1A2 (0.79) MPICYP1A2CYP2C9
SCHEMBL787380 0.73 CYP1A2 (0.67) MPICYP1A2CYP2C9PPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011116356-A2 POSITIVE ALLOSTERIC MODULATORS OF GROUP II MGLURS SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2011-09-22 WO disclosed