SCHEMBL23845

SCHEMBL23845

COc1cccc(C(O)c2cc(Br)cs2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
IGF1R P08069 1/20 0.41
PKM P14618 1/20 0.41
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
BRD4 O60885 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
KDM4A O75164 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
TOP2A P11388 1/20 0.38
TOP2B Q02880 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18529828 0.80 AOC3 (0.50) AOC3L3MBTL1IGF1RPKMCHRM2
SCHEMBL31476413 0.80 AOC3 (0.50) AOC3L3MBTL1IGF1RPKMCHRM2
SCHEMBL12443488 0.79 CNR2 (0.52) AOC3L3MBTL1MEN1KMT2APKM
SCHEMBL2093768 0.79 AOC3 (0.59) AOC3L3MBTL1PKMCHRM2CHRM1
SCHEMBL6598474 0.78 IGF1R (0.50) AOC3L3MBTL1IGF1RPKMCHRM2
SCHEMBL5511034 0.77 TOP2A (0.48) IDO1TOP2ATOP2B
SCHEMBL4822561 0.74 AOC3 (0.54) AOC3L3MBTL1PKMCHRM2CHRM1
SCHEMBL27686957 0.74 AOC3 (0.54) AOC3L3MBTL1PKMCHRM2CHRM1
SCHEMBL477338 0.74 AOC3 (0.54) AOC3L3MBTL1PKMCHRM2CHRM1
SCHEMBL6866452 0.73 AOC3 (0.47) AOC3L3MBTL1PKMCHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed