SCHEMBL23876299

SCHEMBL23876299

Cc1nc(C)c(-c2ccnc(C(C)(C)C)c2)s1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 5/20 0.54
PIK3CD O00329 4/20 0.54
PIK3CB P42338 3/20 0.54
PIK3CG P48736 3/20 0.54
CDK2 P24941 5/20 0.45
CDK4 P11802 4/20 0.45
CCNE1 P24864 1/20 0.45
JAK2 O60674 1/20 0.43
COMT P21964 4/20 0.41
NR2F2 P24468 1/20 0.40
TRPV4 Q9HBA0 2/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
AURKA O14965 1/20 0.38
CDK1 P06493 1/20 0.38
CDK7 P50613 1/20 0.38
CDK9 P50750 1/20 0.38
AURKB Q96GD4 1/20 0.38
PLK1 P53350 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL571475 0.85 PIK3CG (0.52) PIK3CAPIK3CDPIK3CBPIK3CGCDK2
SCHEMBL30476425 0.85 PIK3CG (0.52) PIK3CAPIK3CDPIK3CBPIK3CGCDK2
SCHEMBL18616748 0.82 PIK3CA (0.61) PIK3CAPIK3CDPIK3CBPIK3CGCDK2
SCHEMBL3491367 0.79 PIK3CA (0.55) PIK3CAPIK3CDPIK3CBPIK3CGLMNA
SCHEMBL571448 0.77 PIK3CG (0.71) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL29011650 0.76 PIK3CA (0.55) PIK3CAPIK3CDPIK3CBPIK3CGLMNA
SCHEMBL16045646 0.72 PIK3CA (0.48) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL30500997 0.72 PIK3CA (0.51) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL15801542 0.72 PIK3CA (0.51) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL10145051 0.71 JAK2 (0.45) CDK2CDK4CCNE1JAK2COMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021189143-A1 STABLE HEAVY ISOTOPES IN AMIDE FUNCTIONAL GROUPS AND USES THEREOF Risen (Suzhou) Pharma Tech Co., Ltd. (CN) 2021-09-30 WO disclosed