SCHEMBL23891582

SCHEMBL23891582

C=NCCC1(n2cc(-c3ncnc4[nH]ccc34)cn2)CN(S(=O)(=O)CC)C1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 20/20 0.72
JAK2 O60674 19/20 0.72
JAK3 P52333 15/20 0.72
TYK2 P29597 2/20 0.72
CIT O14578 1/20 0.72
GAK O14976 1/20 0.72
ROCK2 O75116 1/20 0.72
ULK1 O75385 1/20 0.72
PRKCB P05771 1/20 0.72
RET P07949 1/20 0.72
PRKCA P17252 1/20 0.72
PRKACA P17612 1/20 0.72
MARK3 P27448 1/20 0.72
STAT3 P40763 1/20 0.72
CLK1 P49759 1/20 0.72
CSNK1G2 P78368 1/20 0.72
PRKCD Q05655 1/20 0.72
MAP3K1 Q13233 1/20 0.72
ROCK1 Q13464 1/20 0.72
TNK1 Q13470 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23891561 0.91 JAK1 (0.74) JAK1JAK2JAK3TYK2CIT
SCHEMBL17520497 0.88 JAK1 (0.81) JAK1JAK2JAK3TYK2CIT
SCHEMBL13424011 0.87 JAK1 (0.79) JAK1JAK2JAK3TYK2CIT
SCHEMBL872597 0.86 JAK1 (0.78) JAK1JAK2JAK3TYK2CIT
SCHEMBL23557784 0.86 JAK1 (0.72) JAK1JAK2JAK3TYK2CIT
Baricitinib SCHEMBL871150 0.84 JAK1 (1.00) JAK1JAK2JAK3TYK2CIT
Baricitinib SCHEMBL29349824 0.84 JAK1 (1.00) JAK1JAK2JAK3TYK2CIT
SCHEMBL20144680 0.84 JAK1 (1.00) JAK1JAK2JAK3TYK2CIT
SCHEMBL23891585 0.83 JAK1 (0.75) JAK1JAK2JAK3TYK2CIT
Baricitinib SCHEMBL20135561 0.83 JAK1 (0.98) JAK1JAK2JAK3TYK2CIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3728261-B1 CO-CRYSTAL OF AN ORALLY AVAILABLE JANUS KINASE INHIBITOR SANDOZ AG (CH) 2021-10-06 EP disclosed