SCHEMBL23896337

SCHEMBL23896337

CC(=O)NC(C(=O)O)[C@@H](C)Oc1nc(C(C)C)c(-c2ccc(F)cc2)c2ccc(O)c(F)c12

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GCGR P47871 8/20 0.36
MMP1 P03956 1/20 0.31
MMP2 P08253 1/20 0.31
MMP3 P08254 1/20 0.31
MMP7 P09237 1/20 0.31
MMP9 P14780 1/20 0.31
MMP13 P45452 1/20 0.31
ACACB O00763 2/20 0.31
CSGALNACT1 Q8TDX6 1/20 0.31
MAPK13 O15264 1/20 0.31
MAPK12 P53778 1/20 0.31
MAPK11 Q15759 1/20 0.31
MAPK14 Q16539 1/20 0.31
SCN9A Q15858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25545407 1.00 GCGR (0.36) GCGRMMP1MMP2MMP3MMP7
SCHEMBL25543950 1.00 GCGR (0.36) GCGRMMP1MMP2MMP3MMP7
SCHEMBL23887748 0.85 GCGR (0.38) GCGR
SCHEMBL30121089 0.85 GCGR (0.38) GCGR
SCHEMBL25265198 0.85 GCGR (0.38) GCGR
SCHEMBL23896331 0.85 GCGR (0.38) GCGR
SCHEMBL23896334 0.82 GCGR (0.35) GCGR
SCHEMBL25545423 0.78 GCGR (0.43) GCGR
SCHEMBL23896335 0.77 GCGR (0.38) GCGR
SCHEMBL25548631 0.76 GCGR (0.35) GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021203028-A1 7- OR 8-HYDROXY-ISOQUINOLINE AND 7- OR 8-HYDROXY-QUINOLINE DERIVATIVES AS ALPHA-1 -ANTITRYPSIN MODULATORS FOR TREATING ALPHA-1 -ANTITRYPSIN DEFICIENCY (AATD) VERTEX PHARMACEUTICALS INCORPORATED (US) 2021-10-07 WO disclosed