SCHEMBL23918240

SCHEMBL23918240

Cc1nc(Cl)c2cnn(C(C)C)c2n1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
PDE9A O76083 14/20 0.42
KMT2A Q03164 1/20 0.42
PDE1C Q14123 3/20 0.41
PLK4 O00444 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31051051 1.00 KDM4E (0.42) KDM4EPDE9AKMT2APDE1CPLK4
SCHEMBL2357706 0.84 KDM4E (0.43) KDM4EPDE9AKMT2APDE1C
SCHEMBL13251787 0.82 KDM4E (0.44) KDM4EPDE9AKMT2APDE1CPLK4
SCHEMBL31403549 0.81 KDM4E (0.41) KDM4EPDE9AKMT2APDE1CPLK4
SCHEMBL31403622 0.81 ADORA2A (0.46) KDM4EPDE9AKMT2APDE1C
SCHEMBL24500614 0.79 KDM4E (0.42) KDM4EPDE9AKMT2APDE1C
SCHEMBL30095720 0.79 KDM4E (0.40) KDM4EPDE9AKMT2APDE1C
SCHEMBL29174768 0.79 KDM4E (0.40) KDM4EPDE9AKMT2APDE1C
SCHEMBL21282841 0.79 KDM4E (0.40) KDM4EPDE9AKMT2APDE1C
SCHEMBL30095819 0.78 KDM4E (0.50) KDM4EPDE9AKMT2APDE1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117529315-A Imidazole-containing ALK2 kinase inhibitors 生物水晶制药公司 2024-02-06 CN disclosed
EP-3892622-A1 COMPOUNDS HAVING PDE9A INHIBITORY ACTIVITY, AND PHARMACEUTICAL USES THEREOF Korea Research Institute of Chemical Technology (KR) 2021-10-13 EP disclosed