SCHEMBL23922772

SCHEMBL23922772

COc1cc2nccc(Oc3ccc(NC(=O)O)cc3)c2cc1OC

nearest known ligand 0.81

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 15/20 0.81
KDR P35968 13/20 0.81
KIT P10721 1/20 0.76
FLT3 P36888 1/20 0.73
AURKB Q96GD4 1/20 0.73
AXL P30530 1/20 0.72
FGFR2 P21802 2/20 0.70
MET P08581 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27082957 0.91 PDGFRA (0.82) PDGFRAKDRKITFLT3AURKB
SCHEMBL27081475 0.91 PDGFRA (0.95) PDGFRAKDR
SCHEMBL29973354 0.91 PDGFRA (0.95) PDGFRAKDR
SCHEMBL30918281 0.91 PDGFRA (0.82) PDGFRAKDRKITFLT3AURKB
SCHEMBL7490931 0.90 PDGFRA (1.00) PDGFRAKDRKITFGFR2
SCHEMBL6228087 0.89 PDGFRA (0.79) PDGFRAKDRKITFLT3AURKB
SCHEMBL5824534 0.89 PDGFRA (0.79) PDGFRAKDRKITFLT3AURKB
SCHEMBL3931065 0.89 PDGFRA (1.00) PDGFRAKDRFGFR2
SCHEMBL8070553 0.89 PDGFRA (0.94) PDGFRAKDRKIT
SCHEMBL6227250 0.88 PDGFRA (0.85) PDGFRAKDRKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220064117-A1 PAN-KIT KINASE INHIBITOR HAVING QUINOLINE STRUCTURE AND APPLICATION THEREOF Tarapeutics Science Inc. (CN) 2022-03-03 US disclosed
EP-3896059-A1 PAN-KIT KINASE INHIBITOR HAVING QUINOLINE STRUCTURE AND APPLICATION THEREOF Tarapeutics Science Inc. (CN) 2021-10-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220064117-A1 PAN-KIT KINASE INHIBITOR HAVING QUINOLINE STRUCTURE AND APPLICATION THEREOF KIT, MAP3K7, ABL1 PDGFRA 747/4885KDR 357/4885KIT 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.