SCHEMBL23923927

SCHEMBL23923927

Cc1cc2c(NC(=O)C3CN(C(=O)O)CC3c3ccccc3)cccc2cn1

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 18/20 0.44
CYP2D6 P10635 4/20 0.41
CYP3A4 P08684 2/20 0.40
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23923925 1.00 TRPV1 (0.44) TRPV1CYP2D6CYP3A4KDM4E
SCHEMBL23951809 0.88 TACR1 (0.51) TRPV1
SCHEMBL29900568 0.88 TACR1 (0.51) TRPV1
SCHEMBL23924238 0.84 FABP7 (0.55) CYP2D6CYP3A4KDM4E
SCHEMBL23924250 0.84 FABP7 (0.55) CYP2D6CYP3A4KDM4E
SCHEMBL23924239 0.84 FABP7 (0.55) CYP2D6CYP3A4KDM4E
SCHEMBL23924170 0.84 TRPV1 (0.47) TRPV1KDM4E
SCHEMBL23924493 0.84 TRPV1 (0.47) TRPV1KDM4E
SCHEMBL23924172 0.84 TRPV1 (0.47) TRPV1KDM4E
SCHEMBL23924282 0.84 TRPV1 (0.47) TRPV1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115427394-A Heterocyclic compounds for modulating NR2F6 TES制药有限责任公司 2022-12-02 CN disclosed
US-20220213061-A9 HETEROCYCLIC COMPOUNDS FOR MODULATING NR2F6 TES PHARMA S.R.L. (IT) 2022-07-07 US disclosed
US-20210323942-A1 HETEROCYCLIC COMPOUNDS FOR MODULATING NR2F6 TES PHARMA S R L (IT) 2021-10-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220213061-A9 HETEROCYCLIC COMPOUNDS FOR MODULATING NR2F6 NR2E3, NR2F2, NR2C2 TRPV1 4072/4885CYP2D6 2976/4885CYP3A4 4393/4885
US-20210323942-A1 HETEROCYCLIC COMPOUNDS FOR MODULATING NR2F6 NR2E3, NR2F2, NR2C2 TRPV1 4072/4885CYP2D6 2976/4885CYP3A4 4393/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.