SCHEMBL23924495

SCHEMBL23924495

O=C(Nc1cccc2cnccc12)O[C@H]1CN(C(=O)O)C[C@@H]1c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 14/20 0.45
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
BLM P54132 1/20 0.44
ALDH1A1 P00352 3/20 0.41
MAPT P10636 3/20 0.41
KDM4E B2RXH2 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NSD2 O96028 1/20 0.41
LMNA P02545 1/20 0.41
ROCK1 Q13464 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23924496 1.00 TRPV1 (0.45) TRPV1KMT2AMEN1MAPK1HTT
SCHEMBL23924009 0.90 KMT2A (0.48) TRPV1KMT2AMEN1MAPK1HTT
SCHEMBL23924256 0.90 KMT2A (0.48) TRPV1KMT2AMEN1MAPK1HTT
SCHEMBL23924011 0.90 KMT2A (0.48) TRPV1KMT2AMEN1MAPK1HTT
SCHEMBL23951602 0.88 TRPV1 (0.44) TRPV1KMT2AMEN1MAPK1HTT
SCHEMBL23924282 0.83 TRPV1 (0.47) TRPV1KMT2AMEN1MAPK1HTT
SCHEMBL23924170 0.83 TRPV1 (0.47) TRPV1KMT2AMEN1MAPK1HTT
SCHEMBL23924493 0.83 TRPV1 (0.47) TRPV1KMT2AMEN1MAPK1HTT
SCHEMBL23924118 0.83 TRPV1 (0.47) TRPV1KMT2AMEN1MAPK1HTT
SCHEMBL23924172 0.83 TRPV1 (0.47) TRPV1KMT2AMEN1MAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220213061-A9 HETEROCYCLIC COMPOUNDS FOR MODULATING NR2F6 TES PHARMA S.R.L. (IT) 2022-07-07 US disclosed
US-20210323942-A1 HETEROCYCLIC COMPOUNDS FOR MODULATING NR2F6 TES PHARMA S R L (IT) 2021-10-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220213061-A9 HETEROCYCLIC COMPOUNDS FOR MODULATING NR2F6 NR2E3, NR2F2, NR2C2 TRPV1 4072/4885KMT2A 1332/4885MEN1 4081/4885
US-20210323942-A1 HETEROCYCLIC COMPOUNDS FOR MODULATING NR2F6 NR2E3, NR2F2, NR2C2 TRPV1 4072/4885KMT2A 1332/4885MEN1 4081/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.