SCHEMBL2392659

SCHEMBL2392659

CCc1c(C=CC(=O)O)ccc(O)c1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.46
CA1 P00915 4/20 0.45
CA2 P00918 4/20 0.45
CA4 P22748 4/20 0.45
NFKB1 P19838 2/20 0.45
CSNK2A2 P19784 2/20 0.42
CSNK2B P67870 2/20 0.42
CSNK2A1 P68400 2/20 0.42
EIF2AK2 P19525 1/20 0.42
AKR1C3 P42330 2/20 0.41
MIF P14174 1/20 0.41
AKR1C2 P52895 1/20 0.41
KDM4E B2RXH2 5/20 0.40
CA12 O43570 3/20 0.40
CA3 P07451 3/20 0.40
CA6 P23280 3/20 0.40
CA5A P35218 3/20 0.40
CA7 P43166 3/20 0.40
CA9 Q16790 3/20 0.40
CA14 Q9ULX7 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6678566 0.84 ESR1 (0.48) ESR1CA1CA2CA4NFKB1
SCHEMBL2394180 0.84 ESR1 (0.51) ESR1CA1CA2CA4NFKB1
SCHEMBL6668620 0.84 ESR1 (0.48) ESR1CA1CA2CA4NFKB1
SCHEMBL2394170 0.83 MIF (0.46) ESR1CA1CA2CA4NFKB1
SCHEMBL2865033 0.83 CA1 (0.47) ESR1CA1CA2CA4NFKB1
SCHEMBL6855197 0.83 CA1 (0.47) ESR1CA1CA2CA4NFKB1
SCHEMBL2388955 0.83 ESR1 (0.47) ESR1CA1CA2CA4NFKB1
SCHEMBL2389151 0.81 KDM4E (0.47) CA1CA2CA4CSNK2A2CSNK2B
SCHEMBL1405663 0.79 KDM4E (0.46) ESR1CA1CA2CA4NFKB1
SCHEMBL2393450 0.78 ESR1 (0.46) ESR1CA1CA2CA4NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE42700-E1 Induction of apoptosis in cancer cells SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2011-09-13 US disclosed