SCHEMBL23937869

SCHEMBL23937869

Cc1nc(C(F)(F)F)n2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 0.51
PTPN2 P17706 1/20 0.51
SSTR4 P31391 2/20 0.45
HSD17B10 Q99714 1/20 0.39
MAPK1 P28482 1/20 0.38
PRMT6 Q96LA8 1/20 0.38
LMNA P02545 2/20 0.38
TSHR P16473 1/20 0.38
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 1/20 0.37
PDE10A Q9Y233 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20805122 0.84 PTPN1 (0.58) PTPN1PTPN2SSTR4HSD17B10LMNA
SCHEMBL16256059 0.81 PTPN1 (0.50) PTPN1PTPN2SSTR4HSD17B10LMNA
SCHEMBL25527271 0.79 SSTR4 (0.46) PTPN1PTPN2SSTR4HSD17B10MAPK1
SCHEMBL8234959 0.79 PTPN1 (0.60) PTPN1PTPN2SSTR4HSD17B10MAPK1
SCHEMBL20674538 0.79 HSD17B10 (0.39) SSTR4HSD17B10MAPK1LMNATSHR
SCHEMBL23587117 0.76 CYP1A2 (0.42) SSTR4HSD17B10MAPK1KDM4EALDH1A1
SCHEMBL937960 0.75 SSTR4 (0.48) SSTR4HSD17B10MAPK1LMNATSHR
SCHEMBL7499354 0.73 PTGS1 (0.45) SSTR4HSD17B10MAPK1HPGD
SCHEMBL7373417 0.73 CYP1A2 (0.40) SSTR4LMNAKDM4EALDH1A1KMT2A
SCHEMBL20654279 0.72 SSTR4 (0.37) SSTR4HSD17B10MAPK1LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3399968-B1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LTD (KY) 2021-10-20 EP disclosed