SCHEMBL23950303

SCHEMBL23950303

CSNCC(C)n1cnc2c(-c3cccnc3)nc(-c3ccc(N4CCOCC4)cc3)cc2c1=O

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.42
ACVR1 Q04771 1/20 0.40
SYK P43405 12/20 0.40
AURKA O14965 3/20 0.38
PIM1 P11309 1/20 0.37
MTOR P42345 1/20 0.37
MAPK8 P45983 1/20 0.37
MAPK10 P53779 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23950301 0.89 ATR (0.41) ATRACVR1SYKAURKAPIM1
SCHEMBL23925568 0.89 ATR (0.41) ATRACVR1SYKAURKA
SCHEMBL23950770 0.88 ATR (0.44) ATRACVR1SYKAURKAPIM1
SCHEMBL23950297 0.88 ATR (0.44) ATRACVR1SYKPIM1
SCHEMBL23950302 0.87 PSD (0.36) ATRMTOR
SCHEMBL23950547 0.84 SYK (0.43) ATRACVR1SYKAURKAPIM1
SCHEMBL23951143 0.81 SYK (0.45) ATRACVR1SYKAURKAPIM1
SCHEMBL23951142 0.78 SYK (0.47) ATRACVR1SYKAURKAPIM1
SCHEMBL23390302 0.76 CYP2A6 (0.39) PIM1
SCHEMBL23390306 0.76 CYP2A6 (0.39) PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021210970-A1 PYRIDOPYRIMIDINONE DERIVATIVES AND THEIR USE AS ARYL HYDROCARBON RECEPTOR MODULATORS DONG-A ST CO., LTD. (KR) 2021-10-21 WO disclosed