SCHEMBL23950665

SCHEMBL23950665

O=c1c2cc(-c3ccc(C(F)(F)F)cc3)nc(-c3cccnc3)c2ncn1C1CCCCC1O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.51
ALOX5 P09917 1/20 0.42
CHRM1 P11229 1/20 0.42
CYP2C9 P11712 1/20 0.42
PIM1 P11309 1/20 0.36
CYP11B1 P15538 2/20 0.36
TRPV3 Q8NET8 5/20 0.35
HTR2B P41595 1/20 0.35
HTR6 P50406 1/20 0.35
CYP11B2 P19099 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
XBP1 P17861 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
VCP P55072 1/20 0.35
TOP1 P11387 1/20 0.35
GRM2 Q14416 1/20 0.35
SCN9A Q15858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23925444 1.00 KCNH2 (0.51) KCNH2ALOX5CHRM1CYP2C9PIM1
SCHEMBL23925562 1.00 KCNH2 (0.51) KCNH2ALOX5CHRM1CYP2C9PIM1
SCHEMBL23925516 0.89 KCNH2 (0.54) KCNH2ALOX5CHRM1CYP2C9PIM1
SCHEMBL25463136 0.89 KCNH2 (0.54) KCNH2ALOX5CHRM1CYP2C9PIM1
SCHEMBL23950996 0.89 KCNH2 (0.54) KCNH2ALOX5CHRM1CYP2C9PIM1
SCHEMBL25463193 0.89 ACVR1 (0.40) KCNH2PIM1CYP11B1HTR2BHTR6
SCHEMBL23950995 0.87 HTR2B (0.40) KCNH2PIM1CYP11B1HTR2BHTR6
SCHEMBL25463934 0.87 HTR2B (0.40) KCNH2PIM1CYP11B1HTR2BHTR6
SCHEMBL23925713 0.86 CYP11B1 (0.39) KCNH2PIM1CYP11B1HTR2BHTR6
SCHEMBL23951140 0.86 CYP11B1 (0.39) KCNH2PIM1CYP11B1HTR2BHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021210970-A1 PYRIDOPYRIMIDINONE DERIVATIVES AND THEIR USE AS ARYL HYDROCARBON RECEPTOR MODULATORS DONG-A ST CO., LTD. (KR) 2021-10-21 WO disclosed