SCHEMBL23958425

SCHEMBL23958425

CC(C)(F)CN1CCc2cc(OS(=O)(=O)C(F)(F)F)ccc2C1c1ccc(NC2CN(CCCF)C2)cn1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 20/20 0.49
KCNH2 Q12809 11/20 0.49
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45
HDAC6 Q9UBN7 2/20 0.41
HDAC1 Q13547 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958417 0.94 ESR1 (0.48) ESR1KCNH2CYP3A4CYP2D6HRH3
SCHEMBL23958505 0.87 ESR1 (0.52) ESR1KCNH2CYP3A4CYP2D6HRH3
SCHEMBL30211143 0.86 ESR1 (0.63) ESR1KCNH2CYP3A4CYP2D6HRH3
SCHEMBL30822536 0.82 ESR1 (0.63) ESR1KCNH2CYP3A4CYP2D6HRH3
SCHEMBL21583964 0.82 ESR1 (0.63) ESR1KCNH2CYP3A4CYP2D6HRH3
SCHEMBL27105447 0.82 ESR1 (0.63) ESR1KCNH2CYP3A4CYP2D6HRH3
SCHEMBL23929167 0.82 ESR1 (0.63) ESR1KCNH2CYP3A4CYP2D6HRH3
SCHEMBL23958533 0.81 ESR1 (0.51) ESR1KCNH2CYP3A4CYP2D6HRH3
SCHEMBL23958466 0.79 ESR1 (0.49) ESR1KCNH2CYP3A4CYP2D6HRH3
SCHEMBL23958431 0.79 ESR1 (0.44) ESR1KCNH2CYP3A4CYP2D6HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021213358-A1 BORON-CONTAINING COMPOUNDS AND APPLICATION THEREOF 江苏先声药业有限公司 (CN) 2021-10-28 WO disclosed