SCHEMBL23958875

SCHEMBL23958875

COc1cc(C(=O)NCC(c2cc(C(C)(C)O)cc(-c3ccc(F)cc3)n2)C2CC2)cc2cc(C)nnc12

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 6/20 0.36
ABCB1 P08183 1/20 0.34
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
ACSS2 Q9NR19 1/20 0.33
ACACB O00763 1/20 0.32
ACACA Q13085 1/20 0.32
VCP P55072 1/20 0.32
KCNH2 Q12809 1/20 0.32
ALDH1A1 P00352 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MAPT P10636 1/20 0.31
TLR9 Q9NR96 1/20 0.31
TLR8 Q9NR97 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
NR1I2 O75469 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25687466 0.82 SCN9A (0.36) SCN9AABCB1ACACBACACA
SCHEMBL30007220 0.82 SCN9A (0.36) SCN9AABCB1ACACBACACA
SCHEMBL25687467 0.82 SCN9A (0.36) SCN9AABCB1ACACBACACA
SCHEMBL28909130 0.82 SCN9A (0.36) SCN9AABCB1ACACBACACA
SCHEMBL25687476 0.80 SCN9A (0.38) SCN9ATP53ALDH1A1SMN1; SMN2MAPT
SCHEMBL25687377 0.80 SCN9A (0.38) SCN9ATP53ALDH1A1SMN1; SMN2MAPT
SCHEMBL30007116 0.80 SCN9A (0.38) SCN9ATP53ALDH1A1SMN1; SMN2MAPT
SCHEMBL23958713 0.80 SCN9A (0.38) SCN9ATP53ALDH1A1SMN1; SMN2MAPT
SCHEMBL25687474 0.80 SCN9A (0.38) SCN9ATP53ALDH1A1SMN1; SMN2MAPT
SCHEMBL30006910 0.79 SCN9A (0.38) SCN9ATP53ALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed