SCHEMBL2396372

SCHEMBL2396372

N[C@@H](COc1ccc(Cl)cc1)c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SCN4A P35499 10/20 1.00
TACR1 P25103 1/20 0.53
PPARG P37231 1/20 0.50
PPARA Q07869 1/20 0.50
IDO1 P14902 2/20 0.46
TDO2 P48775 2/20 0.46
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA7 P43166 1/20 0.45
CA9 Q16790 1/20 0.45
CYP1A2 P05177 1/20 0.44
DRD2 P14416 1/20 0.44
DRD4 P21917 1/20 0.44
DRD3 P35462 1/20 0.44
CYP19A1 P11511 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15326792 1.00 SCN4A (1.00) SCN4ATACR1PPARGPPARAIDO1
SCHEMBL4345367 0.87 SCN4A (1.00) SCN4ATACR1
SCHEMBL12847267 0.87 SCN4A (1.00) SCN4ATACR1
SCHEMBL12266575 0.82 SCN4A (0.76) SCN4ATACR1CA12CA1CA2
SCHEMBL15326789 0.82 SCN4A (0.76) SCN4ATACR1CYP1A2
SCHEMBL1496649 0.79 SCN4A (0.65) SCN4APPARGPPARACYP1A2
SCHEMBL19686196 0.79 SCN4A (0.76) SCN4A
SCHEMBL19685926 0.77 SCN4A (0.68) SCN4ATACR1
SCHEMBL2397106 0.76 SCN4A (0.61) SCN4ATACR1IDO1TDO2CYP1A2
SCHEMBL3441819 0.76 SCN4A (0.61) SCN4APPARGPPARACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8012901-B1 Method of synthesizing enantiopure mexiletine analogues and novel β-thiophenoxy and pyridyl ethers NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-09-06 US disclosed
US-8012901-B1 Method of synthesizing enantiopure mexiletine analogues and novel β-thiophenoxy and pyridyl ethers NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-09-06 US disclosed
US-8012901-B1 Method of synthesizing enantiopure mexiletine analogues and novel β-thiophenoxy and pyridyl ethers NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-09-06 US disclosed