SCHEMBL23966530

SCHEMBL23966530

CCOC(=O)Cn1nc(Cc2nc3cc(OC)c(Cl)cc3[nH]2)c2ccccc2c1=O

nearest known ligand 0.82

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 12/20 0.82
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
GAA P10253 1/20 0.46
RECQL P46063 1/20 0.45
TP53 P04637 1/20 0.44
ALDH1A1 P00352 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23966531 0.92 S1PR2 (0.87) S1PR2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL23966542 0.91 S1PR2 (0.82) S1PR2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL23908982 0.91 S1PR2 (1.00) S1PR2TP53
SCHEMBL23914603 0.89 S1PR2 (0.81) S1PR2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL23908951 0.85 S1PR2 (1.00) S1PR2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL23914693 0.85 S1PR2 (0.82) S1PR2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL23908889 0.82 S1PR2 (0.93) S1PR2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL23915204 0.81 S1PR2 (0.77) S1PR2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL23914706 0.81 S1PR2 (0.82) S1PR2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL23908925 0.80 S1PR2 (1.00) S1PR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3649119-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS GALAPAGOS NV (BE) 2021-11-03 EP disclosed