SCHEMBL23966568

SCHEMBL23966568

C=CCC(F)COc1cc2[nH]c(Cc3nn(CC(=O)N4CCOCC4)c(=O)c4cc(OC)ccc34)nc2cc1Cl

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 9/20 0.61
PIK3CD O00329 1/20 0.38
PIK3CB P42338 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.34
BRS3 P32247 1/20 0.34
GAA P10253 1/20 0.34
ATM Q13315 1/20 0.34
MEN1 O00255 1/20 0.33
PSMD14 O00487 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
IDH1 O75874 1/20 0.33
RHEB Q15382 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23908996 0.93 S1PR2 (0.67) S1PR2PIK3CDPIK3CBABCG2BRS3
SCHEMBL23908755 0.91 S1PR2 (0.68) S1PR2PIK3CDPIK3CBABCG2BRS3
SCHEMBL23908842 0.83 S1PR2 (0.79) S1PR2GAAMEN1KMT2A
SCHEMBL23908735 0.83 S1PR2 (0.66) S1PR2PIK3CDPIK3CBRHEBNPC1
SCHEMBL23908851 0.82 S1PR2 (0.64) S1PR2IDH1RHEBNPC1RAB9A
SCHEMBL23908912 0.81 S1PR2 (0.80) S1PR2MEN1KMT2A
SCHEMBL23908835 0.81 S1PR2 (0.66) S1PR2GAAATMMEN1ALDH1A1
SCHEMBL23914869 0.80 S1PR2 (0.72) S1PR2PIK3CDPIK3CBMEN1KMT2A
SCHEMBL23908971 0.79 S1PR2 (0.94) S1PR2MEN1ALDH1A1KMT2A
SCHEMBL23908959 0.79 S1PR2 (0.80) S1PR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3649119-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS GALAPAGOS NV (BE) 2021-11-03 EP disclosed