SCHEMBL23966642

SCHEMBL23966642

N#Cc1cc2nc(Cc3nn(CC(=O)N4CCCC4)c(=O)c4ccccc34)[nH]c2cc1OCC(F)F

nearest known ligand 0.63

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 9/20 0.63
KDM4E B2RXH2 2/20 0.39
HSD17B10 Q99714 1/20 0.39
ALDH1A1 P00352 1/20 0.38
MAPT P10636 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
POLB P06746 2/20 0.37
GAA P10253 1/20 0.36
TP53 P04637 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23908890 0.94 S1PR2 (0.66) S1PR2KDM4EHSD17B10ALDH1A1MAPT
SCHEMBL23908781 0.93 S1PR2 (0.60) S1PR2KDM4EHSD17B10MAPTSMN1; SMN2
SCHEMBL23908871 0.93 S1PR2 (0.60) S1PR2KDM4EHSD17B10MAPTSMN1; SMN2
SCHEMBL23908861 0.91 S1PR2 (0.76) S1PR2
SCHEMBL23914585 0.91 S1PR2 (0.68) S1PR2KDM4EHSD17B10ALDH1A1MAPT
SCHEMBL23908790 0.90 S1PR2 (0.61) S1PR2KDM4EHSD17B10MAPTSMN1; SMN2
SCHEMBL23908736 0.90 S1PR2 (0.61) S1PR2KDM4EHSD17B10MAPTSMN1; SMN2
SCHEMBL23909009 0.89 S1PR2 (0.57) S1PR2KDM4EHSD17B10POLBTP53
SCHEMBL23908910 0.89 S1PR2 (0.61) S1PR2KDM4EHSD17B10ALDH1A1MAPT
SCHEMBL23908878 0.89 S1PR2 (0.64) S1PR2KDM4EHSD17B10MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3649119-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS GALAPAGOS NV (BE) 2021-11-03 EP disclosed