SCHEMBL23966872

SCHEMBL23966872

CCOc1cc2[nH]c(Cc3nn(CC)c(=O)c4ccccc34)nc2cc1C(F)(F)F

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 11/20 0.62
AKR1B1 P15121 3/20 0.42
RECQL P46063 1/20 0.41
MAPT P10636 1/20 0.39
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CACNA1H O95180 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23908799 0.88 S1PR2 (0.80) S1PR2AKR1B1CYP1A2CYP3A4CYP2C9
SCHEMBL23909054 0.85 S1PR2 (0.78) S1PR2AKR1B1MAPT
SCHEMBL23914856 0.84 S1PR2 (0.68) S1PR2AKR1B1CYP1A2CYP3A4CYP2C9
SCHEMBL23913415 0.80 S1PR2 (0.94) S1PR2AKR1B1
SCHEMBL23908889 0.78 S1PR2 (0.93) S1PR2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL23909034 0.78 S1PR2 (0.81) S1PR2AKR1B1CYP1A2CYP3A4CYP2C9
SCHEMBL23908800 0.77 S1PR2 (1.00) S1PR2AKR1B1
SCHEMBL23908951 0.76 S1PR2 (1.00) S1PR2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL23908767 0.76 S1PR2 (0.75) S1PR2MAPTCYP1A2CYP3A4CYP2C9
SCHEMBL23915576 0.76 S1PR2 (0.67) S1PR2AKR1B1CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3649119-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS GALAPAGOS NV (BE) 2021-11-03 EP disclosed