SCHEMBL23966878

SCHEMBL23966878

N#Cc1cc2[nH]c(Cc3nn(CC4CCCN4CC(=O)C4CCC4)c(=O)c4ccccc34)nc2cc1OCC(F)F

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 8/20 0.56
HRH1 P35367 12/20 0.39
ADRA1A P35348 9/20 0.39
ADRA1B P35368 9/20 0.39
KCNH2 Q12809 7/20 0.39
HRH3 Q9Y5N1 4/20 0.38
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP2D6 P10635 1/20 0.37
HRH2 P25021 1/20 0.37
HTR2B P41595 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23908928 0.93 S1PR2 (0.63) S1PR2HRH1ADRA1AADRA1BKCNH2
SCHEMBL23966877 0.83 S1PR2 (0.65) S1PR2HRH1ADRA1AADRA1BKCNH2
SCHEMBL23909089 0.83 S1PR2 (0.78) S1PR2CYP3A4CYP2C9CYP2C19
SCHEMBL23908809 0.83 S1PR2 (0.59) S1PR2
SCHEMBL23908802 0.82 S1PR2 (0.56) S1PR2HRH1ADRA1AADRA1BHRH3
SCHEMBL23908736 0.82 S1PR2 (0.61) S1PR2
SCHEMBL23915560 0.81 S1PR2 (0.57) S1PR2
SCHEMBL23908829 0.81 S1PR2 (0.57) S1PR2
SCHEMBL23908878 0.81 S1PR2 (0.64) S1PR2
SCHEMBL23908861 0.80 S1PR2 (0.76) S1PR2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3649119-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS GALAPAGOS NV (BE) 2021-11-03 EP disclosed