SCHEMBL23967004

SCHEMBL23967004

O=C1CCCN1c1cccc(I)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.48
HTR3E A5X5Y0 1/20 0.46
HTR3B O95264 1/20 0.46
HTR3A P46098 1/20 0.46
HTR3D Q70Z44 1/20 0.46
HTR3C Q8WXA8 1/20 0.46
CNR2 P34972 1/20 0.43
ALDH1A1 P00352 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.42
CYP2C19 P33261 1/20 0.42
PDE10A Q9Y233 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PIM1 P11309 2/20 0.39
PIM3 Q86V86 2/20 0.39
PIM2 Q9P1W9 2/20 0.39
MAP4K1 Q92918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20687962 0.81 PARP1 (0.49) PARP1CNR2ALDH1A1CYP1A2CYP3A4
SCHEMBL29464219 0.80 PARP1 (0.48) PARP1CNR2ALDH1A1CYP1A2CYP3A4
SCHEMBL19994372 0.80 PARP1 (0.48) PARP1CNR2ALDH1A1CYP1A2CYP3A4
SCHEMBL20153301 0.80 RECQL (0.60) PARP1HTR3EHTR3BHTR3AHTR3D
SCHEMBL20688055 0.80 PARP1 (0.45) PARP1CNR2ALDH1A1CYP1A2CYP3A4
SCHEMBL22136195 0.78 PARP1 (0.58) PARP1CNR2ALDH1A1CYP1A2CYP3A4
SCHEMBL25364537 0.77 PARP1 (0.48) PARP1CNR2ALDH1A1CYP1A2CYP3A4
SCHEMBL20889900 0.76 PARP1 (0.45) PARP1CNR2ALDH1A1CYP1A2CYP3A4
SCHEMBL536720 0.76 PARP1 (0.57) PARP1CNR2ALDH1A1CYP1A2CYP3A4
SCHEMBL17144056 0.76 ALDH1A1 (0.52) PARP1CNR2ALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3572413-B1 1,2-DIHYDRO-3H-PYRAZOLO[3,4-D]PYRIMIDIN-3-ONE DERIVATIVE AS WEE1 INHIBITOR SHIJIAZHUANG SAGACITY NEW DRUG DEV CO LTD (CN) 2021-11-03 EP disclosed