SCHEMBL23970930

SCHEMBL23970930

CC(C)(C)OC(=O)N1CCCC(NC(=O)c2cc([N+](=O)[O-])c(NCCC(N)=O)cc2F)C1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 7/20 0.45
PARP1 P09874 2/20 0.43
SCN9A Q15858 1/20 0.42
HDAC4 P56524 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
RIPK1 Q13546 1/20 0.40
ANO1 Q5XXA6 2/20 0.39
PBK Q96KB5 1/20 0.38
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
BTK Q06187 1/20 0.38
FPR3 P25089 1/20 0.37
FPR2 P25090 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23970928 0.90 USP30 (0.47) USP30PARP1SCN9AHDAC4HDAC6
SCHEMBL23970663 0.89 USP30 (0.45) USP30PARP1SCN9AHDAC4HDAC6
SCHEMBL23971296 0.88 USP30 (0.44) USP30PARP1SCN9AHDAC4HDAC6
SCHEMBL23970657 0.88 USP30 (0.44) USP30PARP1SCN9AHDAC4HDAC6
SCHEMBL23971294 0.88 USP30 (0.44) USP30PARP1SCN9AHDAC4HDAC6
SCHEMBL30159239 0.88 USP30 (0.41) USP30PARP1SCN9ARIPK1BTK
SCHEMBL23970660 0.88 USP30 (0.44) USP30PARP1SCN9AHDAC4HDAC6
SCHEMBL23970924 0.87 USP30 (0.49) USP30PARP1SCN9AHDAC4HDAC6
SCHEMBL23970662 0.87 USP30 (0.49) USP30PARP1SCN9AHDAC4HDAC6
SCHEMBL23970931 0.87 USP30 (0.44) USP30PARP1SCN9AHDAC4HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222353-A1 MACROCYCLIC INHIBITORS OF PEPTIDYLARGININE DEIMINASES GILEAD SCIENCES, INC. (US) 2021-11-04 WO disclosed