SCHEMBL23970940

SCHEMBL23970940

COC(=O)c1cc(N)c(N)c(F)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.51
ALDH1A1 P00352 7/20 0.51
MAPT P10636 6/20 0.51
HPGD P15428 5/20 0.51
GAA P10253 4/20 0.51
HSD17B10 Q99714 2/20 0.51
GLA P06280 1/20 0.51
CASP1 P29466 1/20 0.51
CASP7 P55210 1/20 0.51
ATM Q13315 1/20 0.51
L3MBTL1 Q9Y468 4/20 0.50
LMNA P02545 3/20 0.50
POLB P06746 2/20 0.50
NFKB1 P19838 1/20 0.50
XDH P47989 1/20 0.50
GFER P55789 1/20 0.50
NFKB2 Q00653 1/20 0.50
RELA Q04206 1/20 0.50
FUT7 Q11130 1/20 0.50
TDP1 Q9NUW8 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3445770 0.90 HDAC1 (0.57) KDM4EALDH1A1MAPTHPGDGAA
SCHEMBL28461177 0.86 KDM4E (0.60) KDM4EALDH1A1MAPTHPGDGAA
SCHEMBL30273152 0.85 KDM4E (0.51) KDM4EALDH1A1MAPTHPGDGAA
SCHEMBL1727263 0.85 KDM4E (0.51) KDM4EALDH1A1MAPTHPGDGAA
SCHEMBL448918 0.84 KDM4E (0.50) KDM4EALDH1A1MAPTHPGDGAA
SCHEMBL752914 0.84 KDM4E (0.58) KDM4EALDH1A1MAPTHPGDGAA
SCHEMBL22642968 0.84 KDM4E (0.48) KDM4EALDH1A1MAPTHPGDGAA
SCHEMBL30152820 0.84 KDM4E (0.58) KDM4EALDH1A1MAPTHPGDGAA
SCHEMBL31701857 0.84 KDM4E (0.48) KDM4EALDH1A1MAPTHPGDGAA
SCHEMBL29878715 0.84 KDM4E (0.50) KDM4EALDH1A1MAPTHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024029489-A1 KIT INHIBITORS, COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF MODULUS DISCOVERY, INC. (JP) 2024-02-08 WO disclosed
WO-2021222353-A1 MACROCYCLIC INHIBITORS OF PEPTIDYLARGININE DEIMINASES GILEAD SCIENCES, INC. (US) 2021-11-04 WO disclosed