SCHEMBL23976342

SCHEMBL23976342

OC[C@@H]1CCCc2c1ccnc2Cl

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 4/20 0.31
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
CYP11B1 P15538 2/20 0.30
CYP11B2 P19099 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28970181 1.00 KDM4C (0.31) KDM4CESR1ESR2CYP11B1CYP11B2
SCHEMBL28970231 1.00 KDM4C (0.31) KDM4CESR1ESR2CYP11B1CYP11B2
SCHEMBL30062822 1.00 KDM4C (0.31) KDM4CESR1ESR2CYP11B1CYP11B2
SCHEMBL23977108 0.78 KDM4C (0.34) KDM4C
SCHEMBL28970161 0.78 KDM4C (0.34) KDM4C
SCHEMBL23987302 0.77 KDM4C (0.31) KDM4C
SCHEMBL24542984 0.72 HTR2A (0.38) KDM4CESR1ESR2CYP11B1CYP11B2
SCHEMBL29673168 0.72 HTR2A (0.38) KDM4CESR1ESR2CYP11B1CYP11B2
SCHEMBL30047508 0.71 CYP11B1 (0.34) CYP11B1CYP11B2
SCHEMBL7776691 0.69 ESR1 (0.53) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220401422-A1 COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF HIF2-alpha AND THEIR METHODS OF USE NOVARTIS AG (CH) 2022-12-22 US disclosed
CN-115485275-A Compounds and compositions that inhibit HIF 2-alpha activity and methods of use thereof 诺华股份有限公司 2022-12-16 CN disclosed
WO-2021217508-A1 COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF HIF2α AND THEIR METHODS OF USE NOVARTIS AG (CH) 2021-11-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220401422-A1 COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF HIF2-alpha AND THEIR METHODS OF USE HIF1AN, HIF1A, EGLN2 KDM4C 1386/4885ESR1 2196/4885ESR2 99/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.