SCHEMBL2397725

SCHEMBL2397725

O[C@H]1CC[C@H](Nc2cccc(Nc3nc4ccc(-c5ccccc5)nc4s3)n2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 14/20 0.50
LCK P06239 12/20 0.49
AURKB Q96GD4 12/20 0.49
BTK Q06187 3/20 0.41
EGFR P00533 1/20 0.41
INSR P06213 1/20 0.41
SRC P12931 1/20 0.41
TEC P42680 1/20 0.41
TXK P42681 1/20 0.41
BMX P51813 1/20 0.41
LRRK2 Q5S007 1/20 0.41
CAMKK2 Q96RR4 1/20 0.41
IRAK4 Q9NWZ3 1/20 0.41
CCNT1 O60563 1/20 0.38
PIM2 Q9P1W9 1/20 0.37
ADORA3 P0DMS8 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA2B P29275 1/20 0.36
ADORA1 P30542 1/20 0.36
HCK P08631 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2397731 1.00 ITK (0.50) ITKLCKAURKBBTKEGFR
SCHEMBL12291553 0.89 NPC1 (0.46) ITKLCKAURKBBTKADORA2A
SCHEMBL2395099 0.87 ITK (0.43) ITKLCKAURKBBTKEGFR
SCHEMBL2395088 0.87 ITK (0.43) ITKLCKAURKBBTKEGFR
SCHEMBL2370861 0.84 ITK (0.49) ITKLCKAURKBBTKEGFR
SCHEMBL2370869 0.84 ITK (0.49) ITKLCKAURKBBTKEGFR
SCHEMBL2396976 0.83 PIK3CG (0.49) ITKLCKAURKBEGFRINSR
SCHEMBL2396989 0.83 PIK3CG (0.49) ITKLCKAURKBEGFRINSR
SCHEMBL2396679 0.81 ITK (0.57) ITKLCKAURKBBTKEGFR
SCHEMBL2396683 0.81 ITK (0.57) ITKLCKAURKBBTKEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011110575-A1 DERIVATIVES OF 2-[2-(BENZO- OR PYRIDO-) THIAZOLYLAMINO]-6-AMINOPYRIDINE, USEFUL IN THE TREATMENT OF RESPIRATORIC, ALLERGIC OR INFLAMMATORY DISEASES GLAXO GROUP LIMITED (GB) 2011-09-15 WO disclosed