SCHEMBL23978024

SCHEMBL23978024

N#Cc1ccnc2sccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 3/20 0.41
CHEK1 O14757 1/20 0.41
AURKA O14965 1/20 0.41
DAPK3 O43293 1/20 0.41
JAK2 O60674 1/20 0.41
MAP4K4 O95819 1/20 0.41
ABL1 P00519 1/20 0.41
NTRK1 P04629 1/20 0.41
LCK P06239 1/20 0.41
FYN P06241 1/20 0.41
CSF1R P07333 1/20 0.41
RET P07949 1/20 0.41
IGF1R P08069 1/20 0.41
MET P08581 1/20 0.41
PDGFRB P09619 1/20 0.41
PIM1 P11309 1/20 0.41
FGFR1 P11362 1/20 0.41
PRKACA P17612 1/20 0.41
LTK P29376 1/20 0.41
KDR P35968 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9332246 0.80 CHEK1 (0.41) LRRK2CHEK1AURKADAPK3JAK2
SCHEMBL5519725 0.76 CSNK1A1 (0.38) LRRK2CHEK1AURKADAPK3JAK2
SCHEMBL31674353 0.74 AURKA (0.37) LRRK2CHEK1AURKADAPK3JAK2
SCHEMBL3979877 0.74 CSNK1A1 (0.37) LRRK2CHEK1AURKADAPK3JAK2
SCHEMBL5530019 0.74 MRGPRX1 (0.38) LRRK2CHEK1AURKADAPK3JAK2
SCHEMBL3998036 0.74 AURKA (0.37) LRRK2CHEK1AURKADAPK3JAK2
SCHEMBL4947345 0.74 ABL1 (0.37) LRRK2CHEK1AURKADAPK3JAK2
SCHEMBL5521208 0.74 CHEK1 (0.34) LRRK2CHEK1AURKADAPK3JAK2
SCHEMBL2178694 0.73 LRRK2 (0.46) LRRK2CHEK1MAPK8CLK2LIMK1
SCHEMBL29367767 0.72 KDR (0.42) LRRK2KDRALDH1A1KDM4EMALT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11622970-B2 BCL-2 inhibitors and their use as pharmaceuticals Prelude Therapeutics Incorporation (US) 2023-04-11 US disclosed
US-20210346405-A1 BCL-2 INHIBITORS AND THEIR USE AS PHARMACEUTICALS PRELUDE THERAPEUTICS INCORPORATED 2021-11-11 US disclosed
US-20210346405-A1 BCL-2 INHIBITORS AND THEIR USE AS PHARMACEUTICALS PRELUDE THERAPEUTICS INCORPORATED 2021-11-11 US disclosed
WO-2021222174-A1 BCL-2 INHIBITORS AND THEIR USE AS PHARMACEUTICALS PRELUDE THERAPEUTICS INCORPORATED (US) 2021-11-04 WO disclosed
WO-2021222174-A1 BCL-2 INHIBITORS AND THEIR USE AS PHARMACEUTICALS PRELUDE THERAPEUTICS INCORPORATED (US) 2021-11-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210346405-A1 BCL-2 INHIBITORS AND THEIR USE AS PHARMACEUTICALS BCL2, BCL2L2, BCL2L1 LRRK2 1035/4885CHEK1 790/4885AURKA 3209/4885
US-11622970-B2 BCL-2 inhibitors and their use as pharmaceuticals BCL2, BCL2L2, BCL2L1 LRRK2 1035/4885CHEK1 790/4885AURKA 3209/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.