SCHEMBL23978660

SCHEMBL23978660

Cc1c(Cl)ccc(N(C)c2ncc3ccccc3n2)c1Cl

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.37
NCF1 P14598 1/20 0.34
FGFR4 P22455 1/20 0.32
HTR3A P46098 1/20 0.31
HRH4 Q9H3N8 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
PDE10A Q9Y233 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30336944 0.81 FGFR4 (0.36) CYP1A2FGFR4PTGDR2
SCHEMBL23978659 0.81 FGFR4 (0.36) CYP1A2FGFR4PTGDR2PDE10A
SCHEMBL30336865 0.81 FGFR4 (0.36) CYP1A2FGFR4PTGDR2PDE10A
SCHEMBL23978658 0.81 FGFR4 (0.36) CYP1A2FGFR4PTGDR2
SCHEMBL23979061 0.78 MAPT (0.36) FGFR4
SCHEMBL12003727 0.72 CYP1A2 (0.56) CYP1A2NCF1HTR3AHRH4PDE10A
SCHEMBL31391395 0.72 CYP1A2 (0.56) CYP1A2NCF1HTR3AHRH4PDE10A
SCHEMBL3337226 0.71 CYP1A2 (0.47) CYP1A2NCF1HTR3AHRH4
Hydrochloric Acid SCHEMBL10583130 0.70 CYP1A2 (0.47) CYP1A2NCF1
SCHEMBL26496227 0.69 KMT2A (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed