SCHEMBL23978993

SCHEMBL23978993

O=C(NC[C@@H](NC(=O)c1c(Cl)cc2c(c1Cl)CCN(Cc1ccccc1)C2=O)C(=O)O)NC1CCc2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 15/20 0.44
ICAM1 P05362 15/20 0.44
ITGAL P20701 15/20 0.44
EPHX2 P34913 4/20 0.42
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30279444 1.00 ITGB2 (0.44) ITGB2ICAM1ITGALEPHX2ALDH1A1
SCHEMBL24803248 1.00 ITGB2 (0.44) ITGB2ICAM1ITGALEPHX2ALDH1A1
SCHEMBL26105351 1.00 ITGB2 (0.44) ITGB2ICAM1ITGALEPHX2ALDH1A1
SCHEMBL23978734 1.00 ITGB2 (0.44) ITGB2ICAM1ITGALEPHX2ALDH1A1
SCHEMBL24804798 0.96 ITGB2 (0.48) ITGB2ICAM1ITGALEPHX2
SCHEMBL23978551 0.96 ITGB2 (0.48) ITGB2ICAM1ITGALEPHX2
SCHEMBL26106455 0.96 ITGB2 (0.48) ITGB2ICAM1ITGALEPHX2
SCHEMBL23978556 0.96 ITGB2 (0.43) ITGB2ICAM1ITGALEPHX2
SCHEMBL30279378 0.96 ITGB2 (0.43) ITGB2ICAM1ITGALEPHX2
SCHEMBL24805349 0.96 ITGB2 (0.43) ITGB2ICAM1ITGALEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed