SCHEMBL2400516

SCHEMBL2400516

O=C1OCCN1c1ccc2nc(Nc3cc(CN4CCCCC4)cc(NC4CCC(O)CC4)n3)sc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 13/20 0.46
AURKB Q96GD4 12/20 0.41
LCK P06239 12/20 0.41
EGFR P00533 1/20 0.40
INSR P06213 1/20 0.40
SRC P12931 1/20 0.40
TEC P42680 1/20 0.40
TXK P42681 1/20 0.40
BMX P51813 1/20 0.40
BTK Q06187 1/20 0.40
LRRK2 Q5S007 1/20 0.40
CAMKK2 Q96RR4 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.40
DYRK2 Q92630 2/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
SSTR5 P35346 1/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2400507 1.00 ITK (0.46) ITKAURKBLCKEGFRINSR
SCHEMBL2399268 0.91 ITK (0.42) ITKAURKBLCKEGFRINSR
SCHEMBL2399275 0.91 ITK (0.42) ITKAURKBLCKEGFRINSR
SCHEMBL2400975 0.91 ITK (0.40) ITKAURKBLCKEGFRINSR
SCHEMBL2400981 0.91 ITK (0.40) ITKAURKBLCKEGFRINSR
SCHEMBL2400450 0.90 ITK (0.42) ITKAURKBLCKEGFRINSR
SCHEMBL2400447 0.90 ITK (0.42) ITKAURKBLCKEGFRINSR
SCHEMBL138715 0.88 LCK (0.51) ITKAURKBLCKEGFRINSR
SCHEMBL138714 0.88 LCK (0.51) ITKAURKBLCKEGFRINSR
SCHEMBL2369772 0.87 ITK (0.43) ITKAURKBLCKEGFRINSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011110575-A1 DERIVATIVES OF 2-[2-(BENZO- OR PYRIDO-) THIAZOLYLAMINO]-6-AMINOPYRIDINE, USEFUL IN THE TREATMENT OF RESPIRATORIC, ALLERGIC OR INFLAMMATORY DISEASES GLAXO GROUP LIMITED (GB) 2011-09-15 WO disclosed