SCHEMBL24009012

SCHEMBL24009012

COc1ccc2ncc(C#N)c(C)c2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 3/20 0.56
RAF1 P04049 2/20 0.56
SRC P12931 7/20 0.55
EGFR P00533 3/20 0.52
HPGDS O60760 1/20 0.49
ABL1 P00519 1/20 0.46
BCR P11274 1/20 0.46
PPARG P37231 1/20 0.46
NCOA2 Q15596 1/20 0.46
NCOA1 Q15788 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
NCOA3 Q9Y6Q9 1/20 0.46
PDE4B Q07343 1/20 0.46
NQO1 P15559 1/20 0.45
NMT1 P30419 1/20 0.43
ABCB1 P08183 1/20 0.43
ABCC1 P33527 1/20 0.43
ABCG2 Q9UNQ0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4744297 0.88 MAP2K1 (0.56) MAP2K1RAF1SRCEGFRHPGDS
SCHEMBL3272746 0.84 SRC (0.60) MAP2K1RAF1SRCEGFRHPGDS
SCHEMBL3273442 0.84 MAP2K1 (0.55) MAP2K1RAF1SRCEGFRHPGDS
SCHEMBL28264974 0.84 MAP2K1 (0.55) MAP2K1RAF1SRCEGFRHPGDS
SCHEMBL3272022 0.84 MAP2K1 (0.55) MAP2K1RAF1SRCEGFRHPGDS
SCHEMBL13865282 0.82 POLB (0.47) EGFRNPSR1KDM4EMAPT
SCHEMBL16480634 0.81 MAP2K1 (0.53) MAP2K1RAF1SRCEGFRHPGDS
SCHEMBL26400641 0.81 MAP2K1 (0.53) MAP2K1RAF1SRCEGFRHPGDS
SCHEMBL3273397 0.80 MAP2K1 (0.52) MAP2K1RAF1SRCEGFRHPGDS
SCHEMBL4743752 0.78 SRC (0.62) MAP2K1SRCEGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021225969-A1 IMINO SULFANONE INHIBITORS OF ENPP1 VOLASTRA THERAPEUTICS, INC. (US) 2021-11-11 WO disclosed