SCHEMBL2401253

SCHEMBL2401253

CNC(=O)c1cc(NC(=O)c2ccc(C)c(Nc3nccc(N4C=CC=NC4)n3)c2)cc(N2CCOCC2)c1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LDLR P01130 5/20 0.52
KIT P10721 5/20 0.52
PCSK9 Q8NBP7 5/20 0.52
MAPK14 Q16539 8/20 0.46
PDGFRB P09619 2/20 0.46
BRAF P15056 4/20 0.45
ABL1 P00519 1/20 0.44
SRC P12931 1/20 0.44
CSF1R P07333 1/20 0.43
JAK2 O60674 1/20 0.42
FLT3 P36888 1/20 0.42
HCK P08631 1/20 0.42
NR2C2 P49116 1/20 0.42
BTK Q06187 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2401256 0.84 LDLR (0.52) LDLRKITPCSK9MAPK14PDGFRB
SCHEMBL1656109 0.80 KIT (0.62) LDLRKITPCSK9MAPK14PDGFRB
SCHEMBL6041097 0.75 BMX (0.46) KITMAPK14PDGFRBABL1CSF1R
SCHEMBL19376720 0.73 ABL1 (0.59) LDLRKITPCSK9MAPK14PDGFRB
SCHEMBL6041094 0.73 ABL1 (0.45) KITPDGFRBABL1
SCHEMBL6041086 0.72 KIT (0.66) KITMAPK14PDGFRBBRAFABL1
SCHEMBL6041148 0.69 ABL1 (0.57) PDGFRBABL1SRCJAK2BTK
SCHEMBL6041098 0.69 ABL1 (0.61) MAPK14PDGFRBABL1
SCHEMBL1653887 0.69 ABL1 (0.74) LDLRKITPCSK9MAPK14PDGFRB
SCHEMBL3560393 0.69 ABL1 (0.47) ABL1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110218187-A1 INHIBITORS OF TYROSINE KINASES BREITENSTEIN WERNER 2011-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110218187-A1 INHIBITORS OF TYROSINE KINASES ABL1, BTK, FLT3 LDLR 2348/4885KIT 254/4885PCSK9 1601/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.