Laduviglusib

Laduviglusib

SCHEMBL240280

Cc1c[nH]c(-c2cnc(NCCNc3ccc(C#N)cn3)nc2-c2ccc(Cl)cc2Cl)n1

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 10/20 0.77
CDK1 P06493 3/20 0.77
GSK3A P49840 3/20 0.77
CCNB2 O95067 2/20 0.77
CCNB1 P14635 2/20 0.77
CCNB3 Q8WWL7 2/20 0.77
RPS6KB1 P23443 1/20 0.77
CDK2 P24941 1/20 0.77
LIMK1 P53667 1/20 0.77
TAOK1 Q7L7X3 1/20 0.77
SLK Q9H2G2 1/20 0.77
CLK4 Q9HAZ1 1/20 0.77
CSNK1G1 Q9HCP0 1/20 0.77
IDH1 O75874 2/20 0.40
TMPRSS4 Q9NRS4 1/20 0.36
CNR1 P21554 2/20 0.35
CNR2 P34972 1/20 0.35
ROS1 P08922 1/20 0.33
KDM1A O60341 1/20 0.33
CRHR1 P34998 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Laduviglusib SCHEMBL29838591 1.00 GSK3B (0.77) GSK3BCDK1GSK3ACCNB2CCNB1
Laduviglusib SCHEMBL29381114 1.00 GSK3B (0.77) GSK3BCDK1GSK3ACCNB2CCNB1
Laduviglusib SCHEMBL17165152 0.99 GSK3B (0.76) GSK3BCDK1GSK3ACCNB2CCNB1
SCHEMBL12552315 0.93 GSK3B (0.67) GSK3BCDK1GSK3ACCNB2CCNB1
SCHEMBL5094723 0.92 GSK3B (0.66) GSK3BCDK1GSK3ACCNB2CCNB1
SCHEMBL4398952 0.92 GSK3B (0.65) GSK3BCDK1GSK3ACCNB2CCNB1
SCHEMBL4404427 0.91 GSK3B (0.64) GSK3BCDK1GSK3ACCNB2CCNB1
SCHEMBL20095066 0.90 GSK3B (0.72) GSK3BCDK1GSK3ACCNB2CCNB1
SCHEMBL26489229 0.90 GSK3B (0.62) GSK3BCDK1GSK3ACCNB2CCNB1
SCHEMBL7148131 0.89 GSK3B (0.71) GSK3BCDK1GSK3ACCNB2CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 686 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240352422-A1 DIRECT REPROGRAMMING OF CELLS INTO CARDIAC PURKINJE-LIKE CELLS USING A UNIVERSAL SMALLMOLECULE COCKTAIL UNIVERSITY OF HOUSTON SYSTEM (US) 2024-10-24 US claimed
WO-2024136442-A1 METHOD FOR PREPARING PANCREATIC ISLET ORGANOID USING STATIC SUSPENSION CULTURE METHOD 주식회사 강스템바이오텍 2024-06-27 WO claimed
EP-3384007-B1 IMPROVED METHODS FOR REPROGRAMING NON-PLURIPOTENT CELLS INTO PLURIPOTENT STEM CELLS BEIHAO STEM CELL AND REGENERATIVE MEDICINE RES INSTITUTE CO LTD (CN) 2024-03-27 EP claimed
WO-2023167986-A1 METHODS AND COMPOSITIONS FOR TREATING HEARING LOSS Lineage Cell Therapeutics, Inc. (US) 2023-09-07 WO claimed
US-11655449-B2 Culture conditions to prolong/enhanced endodermal cell type for cell transplantation BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-05-23 US claimed
WO-2023022892-A1 DIRECT REPROGRAMMING OF CELLS INTO CARDIAC PURKINJE-LIKE CELLS USING A UNIVERSAL SMALLMOLECULE COCKTAIL UNIVERSITY OF HOUSTON SYSTEM (US) 2023-02-23 WO claimed
US-20220389376-A1 Methods for Reprogramming Cells NANTES UNIVERSITE (FR) 2022-12-08 US claimed
CN-110564677-B Inducer for inducing pluripotent stem cells to differentiate into beating cardiac muscle cells and application thereof 上海泉生生物科技有限公司 2022-09-09 CN claimed
WO-2021092657-A1 METHODS FOR REPROGRAMMING CELLS MONASH UNIVERSITY (AU) 2021-05-20 WO claimed
US-20210123017-A1 METHOD FOR PRODUCING DOPAMINERGIC NEURONS NATIONAL UNIVERSITY CORPORATION NAGOYA UNIVERSITY (JP) 2021-04-29 US claimed
WO-2013129929-A1 METHODS FOR ACTIVATING RETROVIRUS IN LATENT INFECTED CELLS, AND COMPOUNDS FOR USE THEREIN ERASMUS UNIVERSITY MEDICAL CENTER ROTTERDAM (NL) 2013-09-06 WO claimed
US-20130210060-A1 METHOD OF PRODUCING PANCREATIC HORMONE-PRODUCING CELLS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-08-15 US claimed
WO-2013098140-A1 PERITONEAL DIALYSIS FLUID COMPRISING A GSK-3 INHIBITOR ZYTOPROTEC GMBH (AT) 2013-07-04 WO claimed
EP-2609918-A1 Peritoneal dialysis fluid comprising a GSK-3 inhibitor Zytoprotec GmbH (AT) 2013-07-03 EP claimed
EP-2604685-A1 METHOD OF PRODUCING PANCREATIC HORMONE-PRODUCING CELLS Takeda Pharmaceutical Company Limited (JP) 2013-06-19 EP claimed
US-20130022986-A1 METHOD FOR MANUFACTURING PANCREATIC-HORMONE-PRODUCING CELLS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-01-24 US claimed
US-20120190112-A1 Differentiation of Pluripotent Stem Cells CENTOCOR ORTHO BIOTECH INC. 2012-07-26 US claimed
EP-2283114-A2 TREATMENT OF PLURIPOTENT CELLS Centocor Ortho Biotech Inc. (US) 2011-02-16 EP claimed
US-20090325293-A1 TREATMENT OF PLURIPOTENT CELLS JANSSEN BIOTECH, INC. 2009-12-31 US claimed
WO-2009132068-A2 TREATMENT OF PLURIPOTENT CELLS CENTOCOR ORTHO BIOTECH INC. (US) 2009-10-29 WO claimed