SCHEMBL24035973

SCHEMBL24035973

CCn1c(-c2noc(CNC(=O)c3ccn(C(C)(C)C)c3)n2)cc2c(NC(=O)OC(C)(C)C)cccc21

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.37
THRB P10828 2/20 0.37
KMT2A Q03164 2/20 0.36
CYP2D6 P10635 1/20 0.35
CNR2 P34972 5/20 0.35
HTT P42858 1/20 0.34
TP53 P04637 1/20 0.34
ACSS2 Q9NR19 1/20 0.33
CNR1 P21554 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24852871 0.92 MAPT (0.36) MAPTTHRBKMT2ACYP2D6TP53
SCHEMBL26734850 0.85 MAPT (0.40) MAPTTHRBKMT2ACNR2HTT
SCHEMBL24035966 0.85 MAPT (0.38) MAPTTHRBKMT2ACNR2HTT
SCHEMBL24853071 0.79 MAPT (0.36) MAPTTHRBKMT2ATP53
SCHEMBL26735192 0.79 IRAK4 (0.33) MAPTTHRBCNR2ACSS2CNR1
SCHEMBL24035963 0.79 CNR2 (0.31) MAPTTHRBCNR2TP53CNR1
SCHEMBL26735719 0.78 CYP2D6 (0.41) MAPTTHRBKMT2ACYP2D6CNR2
SCHEMBL24035241 0.78 CYP2D6 (0.43) MAPTCYP2D6CNR2TP53CNR1
SCHEMBL24035888 0.77 MAPT (0.38) MAPTTHRBKMT2AHTTTP53
SCHEMBL24852874 0.77 MAPT (0.37) MAPTTHRBKMT2AHTTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11807644-B2 Methods and compounds for restoring mutant p53 function PMV PHARMACEUTICALS, INC. (US) 2023-11-07 US disclosed
WO-2021231474-A1 METHODS AND COMPOUNDS FOR RESTORING MUTANT p53 FUNCTION PMV PHARMACEUTICALS, INC. (US) 2021-11-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11807644-B2 Methods and compounds for restoring mutant p53 function TP53, TP53BP1, HRAS MAPT 4180/4885THRB 2152/4885KMT2A 3003/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.