SCHEMBL24070548

SCHEMBL24070548

Cc1cn(-c2cc(NC(=O)c3ccc(C)c(CN)c3)cc(C(F)(F)F)c2)cn1

nearest known ligand 0.69

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR2E1 Q9Y466 4/20 0.69
LDLR P01130 1/20 0.67
KIT P10721 1/20 0.67
PCSK9 Q8NBP7 1/20 0.67
ABL1 P00519 8/20 0.67
BCR P11274 7/20 0.67
MAPK14 Q16539 1/20 0.65
MAP3K20 Q9NYL2 1/20 0.65
EPHB2 P29323 1/20 0.65
MAP4K2 Q12851 2/20 0.62
MAP3K7 O43318 1/20 0.61
RAF1 P04049 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30211962 1.00 NR2E1 (0.69) NR2E1LDLRKITPCSK9ABL1
SCHEMBL13659898 0.88 NR2E1 (0.77) NR2E1LDLRKITPCSK9ABL1
SCHEMBL4254144 0.88 NR2E1 (0.73) NR2E1LDLRKITPCSK9ABL1
SCHEMBL28971895 0.88 NR2E1 (0.68) NR2E1LDLRKITPCSK9ABL1
SCHEMBL4254143 0.86 NR2E1 (0.71) NR2E1LDLRKITPCSK9ABL1
SCHEMBL589522 0.86 NR2E1 (0.73) NR2E1LDLRKITPCSK9ABL1
SCHEMBL29493483 0.86 NR2E1 (0.73) NR2E1LDLRKITPCSK9ABL1
SCHEMBL24532047 0.86 NR2E1 (0.73) NR2E1LDLRKITPCSK9ABL1
SCHEMBL24070143 0.85 DDR1 (0.65) NR2E1LDLRKITPCSK9ABL1
SCHEMBL30211927 0.85 DDR1 (0.65) NR2E1LDLRKITPCSK9ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230227447-A1 BENZYLAMINE DERIVATIVES AS DDRS INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2023-07-20 US disclosed
US-20230227447-A1 BENZYLAMINE DERIVATIVES AS DDRS INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2023-07-20 US disclosed
US-20230227447-A1 BENZYLAMINE DERIVATIVES AS DDRS INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2023-07-20 US disclosed
CN-115697485-A Benzylamine derivatives as DDR inhibitors 奇斯药制品公司 2023-02-03 CN disclosed
WO-2021239643-A1 BENZYLAMINE DERIVATIVES AS DDRS INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2021-12-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230227447-A1 BENZYLAMINE DERIVATIVES AS DDRS INHIBITORS DDR2, DDR1, DDRGK1 NR2E1 134/4885LDLR 469/4885KIT 2506/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.