SCHEMBL2409767

SCHEMBL2409767

CN(Cc1c[nH]c(-c2cccnc2F)c1)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.38
SLC6A4 P31645 7/20 0.38
PDK2 Q15119 1/20 0.37
TACR1 P25103 2/20 0.37
CACNA1G O43497 1/20 0.37
CACNA1B Q00975 1/20 0.37
CACNA1C Q13936 1/20 0.37
HTR2A P28223 1/20 0.36
GLS O94925 1/20 0.35
SSTR4 P31391 1/20 0.34
MGLL Q99685 1/20 0.34
HCRTR1 O43613 1/20 0.33
GSK3B P49841 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
RIPK1 Q13546 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2411260 0.86 PLCG1 (0.37) HTR2CSLC6A4PDK2TACR1CACNA1G
SCHEMBL15731438 0.86 HTR2C (0.39) HTR2CSLC6A4PDK2CACNA1GCACNA1B
SCHEMBL5008198 0.84 TACR1 (0.38) TACR1FFAR4
SCHEMBL4430054 0.82 PTGER2 (0.30) HTR2CSLC6A4TACR1RIPK1
SCHEMBL30131039 0.81 HTR2C (0.41) HTR2CSLC6A4PDK2CACNA1GCACNA1B
SCHEMBL1156849 0.81 HTR2C (0.43) HTR2CSLC6A4PDK2CACNA1GCACNA1B
SCHEMBL1156833 0.81 HTR2C (0.41) HTR2CSLC6A4PDK2CACNA1GCACNA1B
SCHEMBL1830977 0.81 SSTR4 (0.38) HTR2CSLC6A4PDK2TACR1CACNA1G
SCHEMBL4566437 0.80 FFAR4 (0.33) TACR1GSK3BFFAR4
SCHEMBL1157177 0.79 SLC6A4 (0.41) HTR2CSLC6A4PDK2CACNA1GCACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed