SCHEMBL2415217

SCHEMBL2415217

CCC(c1ccccc1)c1ccc2oc(-c3ccc(CN4CC(C(=O)O)C4C)cc3F)cc2c1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 17/20 0.53
S1PR3 Q99500 9/20 0.53
KCNH2 Q12809 1/20 0.53
MAOB P27338 3/20 0.46
MAOA P21397 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2420094 0.91 S1PR1 (0.54) S1PR1S1PR3KCNH2MAOBMAOA
SCHEMBL1602190 0.86 S1PR1 (0.71) S1PR1S1PR3KCNH2
SCHEMBL1602087 0.81 S1PR1 (0.61) S1PR1S1PR3KCNH2
SCHEMBL3706281 0.80 S1PR1 (0.52) S1PR1S1PR3KCNH2MAOBMAOA
SCHEMBL1601626 0.79 S1PR1 (0.61) S1PR1S1PR3KCNH2MAOB
SCHEMBL1601723 0.77 S1PR1 (0.73) S1PR1S1PR3KCNH2
SCHEMBL12269426 0.76 S1PR1 (0.74) S1PR1S1PR3KCNH2
SCHEMBL1602358 0.76 S1PR1 (0.74) S1PR1S1PR3KCNH2
SCHEMBL2412108 0.74 S1PR1 (0.50) S1PR1S1PR3KCNH2MAOB
SCHEMBL12269470 0.72 S1PR1 (0.62) S1PR1S1PR3KCNH2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364976-A1 S1P receptor modulating compounds and use thereof EPIX Pharmaceuticals, Inc. (US) 2011-09-14 EP disclosed