SCHEMBL24153992

SCHEMBL24153992

Cc1nc2cncc(Br)c2nc1C

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.39
MAPT P10636 2/20 0.35
PRNP P04156 2/20 0.32
NPSR1 Q6W5P4 2/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32
HTT P42858 1/20 0.32
NOD2 Q9HC29 1/20 0.32
RPS6KA5 O75582 1/20 0.31
ALDH1A1 P00352 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16719118 0.79 PDE10A (0.35) MAPTPRNPHTTALDH1A1RXFP1
SCHEMBL16719083 0.75 CCNB2 (0.30) RPS6KA5
SCHEMBL13348648 0.74 HPGD (0.35) NQO2MAPTPRNPNPSR1LMNA
SCHEMBL24154377 0.74 RPS6KA5 (0.32) RPS6KA5NPC1RAB9AKMT2A
SCHEMBL2513088 0.70 MAPT (0.44) NQO2MAPTPRNPHPGDALDH1A1
SCHEMBL30217623 0.70 MAPT (0.44) NQO2MAPTPRNPHPGDALDH1A1
SCHEMBL27166952 0.67 NQO2 (0.46) NQO2MAPTPRNPNPSR1LMNA
SCHEMBL24153281 0.67 NQO2 (0.45) NQO2MAPTPRNPNPSR1LMNA
SCHEMBL30408222 0.67 NQO2 (0.45) NQO2MAPTPRNPNPSR1LMNA
SCHEMBL31259133 0.66 NQO2 (0.54) NQO2MAPTPRNPNPSR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024109660-A1 CDK INHIBITORS 上海齐鲁制药研究中心有限公司 2024-05-30 WO disclosed
US-20230219934-A1 2,3-DISUBSTITUTED PYRIDO[3,4-B]PYRAZINE-CONTAINING COMPOUNDS AS KINASE INHIBITORS PURDUE RESEARCH FOUNDATION (US) 2023-07-13 US disclosed
US-20230219934-A1 2,3-DISUBSTITUTED PYRIDO[3,4-B]PYRAZINE-CONTAINING COMPOUNDS AS KINASE INHIBITORS PURDUE RESEARCH FOUNDATION (US) 2023-07-13 US disclosed
US-20230219934-A1 2,3-DISUBSTITUTED PYRIDO[3,4-B]PYRAZINE-CONTAINING COMPOUNDS AS KINASE INHIBITORS PURDUE RESEARCH FOUNDATION (US) 2023-07-13 US disclosed
EP-4175957-A1 2,3-DISUBSTITUTED PYRIDO[3,4-B]PYRAZINE-CONTAINING COMPOUNDS AS KINASE INHIBITORS Purdue Research Foundation (US) 2023-05-10 EP disclosed
WO-2021262915-A1 2,3-DISUBSTITUTED PYRIDO[3,4-B]PYRAZINE-CONTAINING COMPOUNDS AS KINASE INHIBITORS PURDUE RESEARCH FOUNDATION (US) 2021-12-30 WO disclosed
WO-2021262915-A1 2,3-DISUBSTITUTED PYRIDO[3,4-B]PYRAZINE-CONTAINING COMPOUNDS AS KINASE INHIBITORS PURDUE RESEARCH FOUNDATION (US) 2021-12-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230219934-A1 2,3-DISUBSTITUTED PYRIDO[3,4-B]PYRAZINE-CONTAINING COMPOUNDS AS KINASE INHIBITORS MAP3K2, MAP4K2, MAP3K5 NQO2 1523/4885MAPT 1649/4885PRNP 1638/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.