SCHEMBL24192811

SCHEMBL24192811

Nc1ccc(CN2CCC(N3CCOCC3)C2)c(C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.53
MAP4K4 O95819 1/20 0.42
PDE3B Q13370 2/20 0.40
PDE3A Q14432 2/20 0.40
DDR1 Q08345 5/20 0.37
CHRM1 P11229 4/20 0.37
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
DRD2 P14416 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24192814 0.84 NR1H2 (0.58) NR1H2DDR1KDM4EALDH1A1
SCHEMBL2435935 0.83 NR1H2 (0.70) NR1H2PDE3BPDE3AKDM4EALDH1A1
SCHEMBL30900087 0.83 NR1H2 (0.70) NR1H2PDE3BPDE3AKDM4EALDH1A1
SCHEMBL15688033 0.81 NR1H2 (0.60) NR1H2CHRM1CCNCCDK8KDM4E
SCHEMBL274890 0.79 NR1H2 (0.69) NR1H2DDR1CHRM1KDM4EALDH1A1
SCHEMBL29958956 0.79 NR1H2 (0.69) NR1H2DDR1CHRM1KDM4EALDH1A1
SCHEMBL27088110 0.79 NR1H2 (0.64) NR1H2PDE3BPDE3ADDR1KDM4E
SCHEMBL24565655 0.78 NR1H2 (0.64) NR1H2PDE3BPDE3AKDM4EALDH1A1
SCHEMBL24192809 0.77 NR1H2 (0.66) NR1H2DDR1CHRM1KDM4EALDH1A1
SCHEMBL15687979 0.76 NR1H2 (0.61) NR1H2MAP4K4DDR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022008383-A1 ISOQUINOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF DISEASES GALAPAGOS NV (BE) 2022-01-13 WO disclosed