SCHEMBL24201824

SCHEMBL24201824

CCNC(=O)/C(C)=N/c1c(C)ncnc1N1CCc2cc(F)ccc21

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 10/20 0.45
MKNK2 Q9HBH9 10/20 0.45
EIF4E P06730 6/20 0.45
NOTUM Q6P988 1/20 0.39
ROCK1 Q13464 1/20 0.36
KIT P10721 1/20 0.35
KCNQ2 O43526 1/20 0.35
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
LMNA P02545 1/20 0.34
SRD5A1 P18405 1/20 0.34
SRD5A2 P31213 1/20 0.34
IDO1 P14902 1/20 0.33
EGFR P00533 1/20 0.33
AKT1 P31749 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23761435 0.90 MKNK1 (0.45) MKNK1MKNK2EIF4ENOTUMROCK1
SCHEMBL23761323 0.89 MKNK1 (0.48) MKNK1MKNK2EIF4ENOTUMROCK1
SCHEMBL23761212 0.88 MKNK1 (0.45) MKNK1MKNK2EIF4ENOTUMKCNQ2
SCHEMBL23761308 0.88 MKNK1 (0.48) MKNK1MKNK2EIF4ENOTUMROCK1
SCHEMBL23761391 0.86 MKNK1 (0.45) MKNK1MKNK2EIF4ENOTUMEGFR
SCHEMBL23761345 0.85 MKNK1 (0.45) MKNK1MKNK2EIF4ENOTUMKIT
SCHEMBL23761515 0.85 MKNK1 (0.45) MKNK1MKNK2EIF4ENOTUMROCK1
SCHEMBL23761447 0.84 MKNK1 (0.41) MKNK1MKNK2EIF4ENOTUMROCK1
SCHEMBL23761492 0.84 MKNK1 (0.45) MKNK1MKNK2EIF4ENOTUMROCK1
SCHEMBL23761495 0.83 MKNK1 (0.55) MKNK1MKNK2EIF4ENOTUMROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3939981-A1 FUSED THIAZOLOPYRIMIDINE DERIVATIVES AS MNKS INHIBITORS LifeArc (GB) 2022-01-19 EP disclosed