SCHEMBL2423819

SCHEMBL2423819

CC(C)[C@H](N[C@H]1CC[C@@H]2CN(S(=O)(=O)c3ccc(C(F)(F)F)cc3)C[C@@H]21)C(N)=O

nearest known ligand 0.68

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 14/20 0.68
GAA P10253 1/20 0.44
EPHX2 P34913 2/20 0.43
MMP1 P03956 1/20 0.43
MMP2 P08253 1/20 0.43
MMP3 P08254 1/20 0.43
MMP7 P09237 1/20 0.43
MMP9 P14780 1/20 0.43
MMP13 P45452 1/20 0.43
TRPV4 Q9HBA0 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16497775 0.91 CACNA1B (0.61) CACNA1BGAAEPHX2TRPV4
SCHEMBL16497772 0.91 CACNA1B (0.61) CACNA1BGAAEPHX2TRPV4
SCHEMBL66757 0.86 CACNA1B (0.74) CACNA1BGAAEPHX2
SCHEMBL2457872 0.85 CACNA1B (0.66) CACNA1BGAAEPHX2
SCHEMBL66019 0.85 CACNA1B (0.66) CACNA1BGAAEPHX2
SCHEMBL3246463 0.85 CACNA1B (0.66) CACNA1BGAAEPHX2
SCHEMBL66747 0.84 CACNA1B (0.74) CACNA1BGAAEPHX2TRPV4
SCHEMBL64800 0.84 CACNA1B (0.77) CACNA1BGAAEPHX2
SCHEMBL66566 0.84 CACNA1B (0.77) CACNA1BGAAEPHX2
SCHEMBL65961 0.84 CACNA1B (0.74) CACNA1BGAAEPHX2TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367790-A2 SUBSTITUTED OCTAHYDROCYCLOPENTA(C)PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS Abbott Laboratories (US) 2011-09-28 EP claimed