SCHEMBL2424490

SCHEMBL2424490

C=CCc1c(OC)cc2c(c1OC)OCO2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 1.00
CYP3A4 P08684 3/20 0.63
ALDH1A1 P00352 2/20 0.63
SMN1; SMN2 Q16637 1/20 0.63
ALOX15 P16050 1/20 0.62
P2RX7 Q99572 2/20 0.44
GSK3B P49841 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ATR Q13535 1/20 0.44
TARBP2 Q15633 1/20 0.43
OPRK1 P41145 1/20 0.42
HTT P42858 1/20 0.42
RECQL P46063 1/20 0.42
LMNA P02545 1/20 0.42
HPGD P15428 1/20 0.42
ACHE P22303 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14552379 0.84 POLB (0.72) POLBCYP3A4ALDH1A1SMN1; SMN2ALOX15
Dillapiole SCHEMBL310992 0.83 POLB (0.71) POLBCYP3A4ALDH1A1SMN1; SMN2ALOX15
SCHEMBL3486950 0.80 POLB (1.00) POLBCYP3A4ALDH1A1SMN1; SMN2ALOX15
SCHEMBL24242264 0.78 POLB (0.64) POLBCYP3A4ALDH1A1SMN1; SMN2ALOX15
SCHEMBL29549259 0.78 POLB (0.63) POLBCYP3A4ALDH1A1SMN1; SMN2ALOX15
Elemicin SCHEMBL30363316 0.78 CYP3A4 (1.00) POLBCYP3A4ALDH1A1SMN1; SMN2ALOX15
Elemicin SCHEMBL68041 0.78 CYP3A4 (1.00) POLBCYP3A4ALDH1A1SMN1; SMN2ALOX15
Elemicin SCHEMBL10728512 0.78 CYP3A4 (1.00) POLBCYP3A4ALDH1A1SMN1; SMN2ALOX15
SCHEMBL14552303 0.77 POLB (0.63) POLBCYP3A4ALDH1A1SMN1; SMN2ALOX15
SCHEMBL14552377 0.77 POLB (0.63) POLBCYP3A4ALDH1A1SMN1; SMN2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090081119-A1 INHIBITING DNA POLYMERASE BETA TO ENHANCE EFFICACY OF ANTICANCER AGENTS UNIVERSITY OF PITTSBURGH-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2009-03-26 US claimed
WO-2007001684-A9 INHIBITING DNA POLYMERASE BETA TO ENHANCE EFFICACY OF ANTICANCER AGENTS UNIV PITTSBURGH (US) 2007-04-19 WO claimed
WO-2007001684-A2 INHIBITING DNA POLYMERASE BETA TO ENHANCE EFFICACY OF ANTICANCER AGENTS UNIVERSITY OF PITTSBURGH OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2007-01-04 WO claimed
CN-109380653-A Preparation method of colorful glutinous rice 谢林峰 2019-02-26 CN disclosed
CN-109247507-A Colorful rice dumpling and preparation method thereof 谢林峰 2019-01-22 CN disclosed
WO-2011112067-A1 A HERBAL COMPOSITION HAVING ANTI-OBESITY PROPERTY UNIVERSITI SAINS MALAYSIA (MY) 2011-09-15 WO disclosed
US-20100048682-A1 INHIBITING DNA POLYMERASE BETA TO ENHANCE EFFICACY OF ANTICANCER AGENTS UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 2010-02-25 US disclosed
US-20090081119-A1 INHIBITING DNA POLYMERASE BETA TO ENHANCE EFFICACY OF ANTICANCER AGENTS UNIVERSITY OF PITTSBURGH-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2009-03-26 US disclosed
WO-2007001684-A9 INHIBITING DNA POLYMERASE BETA TO ENHANCE EFFICACY OF ANTICANCER AGENTS UNIV PITTSBURGH (US) 2007-04-19 WO disclosed
WO-2007001684-A2 INHIBITING DNA POLYMERASE BETA TO ENHANCE EFFICACY OF ANTICANCER AGENTS UNIVERSITY OF PITTSBURGH OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2007-01-04 WO disclosed
US-4876277-A XANTHOMONAS, ERYSIPHE PLANT CELL RESEARCH INSTITUTE, INC. (US) 1989-10-24 US disclosed
US-4803290-A 1,2-AKKYLIDENE DIOXYBENZENE; FUNGICIDES PCRI, INC. (US) 1989-02-07 US disclosed