SCHEMBL24257008

SCHEMBL24257008

C[C@H](N)CNc1nccc(-c2sc(C(C)(C)C)nc2-c2cccc(NS(=O)(=O)c3c(F)cccc3F)c2F)n1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 20/20 0.73
NR1I2 O75469 2/20 0.73
PLK4 O00444 1/20 0.73
EPHB6 O15197 1/20 0.73
RIPK2 O43353 1/20 0.73
JAK2 O60674 1/20 0.73
ULK1 O75385 1/20 0.73
ERN1 O75460 1/20 0.73
PRKD3 O94806 1/20 0.73
ABL1 P00519 1/20 0.73
KRAS P01116 1/20 0.73
RAF1 P04049 1/20 0.73
LCK P06239 1/20 0.73
FYN P06241 1/20 0.73
CDK1 P06493 1/20 0.73
YES1 P07947 1/20 0.73
LYN P07948 1/20 0.73
MET P08581 1/20 0.73
HCK P08631 1/20 0.73
FGR P09769 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30464236 1.00 BRAF (0.73) BRAFNR1I2PLK4EPHB6RIPK2
SCHEMBL12350392 0.94 BRAF (0.73) BRAFNR1I2PLK4EPHB6RIPK2
SCHEMBL1127862 0.92 BRAF (0.73) BRAFNR1I2PLK4EPHB6RIPK2
SCHEMBL27979982 0.92 BRAF (0.73) BRAFNR1I2PLK4EPHB6RIPK2
SCHEMBL2193728 0.92 BRAF (0.73) BRAFNR1I2PLK4EPHB6RIPK2
SCHEMBL19295059 0.90 BRAF (0.77) BRAFNR1I2PLK4EPHB6RIPK2
SCHEMBL19295130 0.90 BRAF (0.70) BRAFNR1I2PLK4EPHB6RIPK2
SCHEMBL12350394 0.88 BRAF (0.76) BRAFNR1I2PLK4EPHB6RIPK2
SCHEMBL20805408 0.88 BRAF (0.81) BRAFNR1I2PLK4EPHB6RIPK2
SCHEMBL24257174 0.88 BRAF (0.70) BRAFNR1I2PLK4EPHB6RIPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230303551-A1 N-CYCLYL-SULFONAMIDES USEFUL FOR INHIBITING RAF ALBERT EINSTEIN COLLEGE OF MEDICINE 2023-09-28 US disclosed
WO-2022036176-A1 N-CYCLYL-SULFONAMIDES USEFUL FOR INHIBITING RAF ALBERT EINSTEIN COLLEGE OF MEDICINE (US) 2022-02-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230303551-A1 N-CYCLYL-SULFONAMIDES USEFUL FOR INHIBITING RAF BRAF, RAF1, NRAS BRAF 1/4885NR1I2 673/4885PLK4 1331/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.