SCHEMBL24257539

SCHEMBL24257539

Cc1c(-c2cccc(Oc3ccccc3)c2)cnc(C(=O)O)c1OCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.44
MRGPRX4 Q96LA9 1/20 0.43
DHODH Q02127 3/20 0.42
P2RX3 P56373 1/20 0.42
PTGER4 P35408 1/20 0.42
NR4A2 P43354 2/20 0.41
ALKBH1 Q13686 1/20 0.41
FFAR1 O14842 4/20 0.41
FFAR4 Q5NUL3 2/20 0.41
PTGER1 P34995 1/20 0.41
MAOB P27338 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Glycine SCHEMBL29248949 0.95 MCL1 (0.41) MCL1MRGPRX4DHODHP2RX3PTGER4
SCHEMBL24257685 0.91 MAOB (0.47) MRGPRX4DHODHPTGER4MAOB
SCHEMBL30453121 0.91 MAOB (0.47) MRGPRX4DHODHPTGER4MAOB
SCHEMBL24257668 0.88 FFAR1 (0.43) MRGPRX4DHODHPTGER4FFAR1FFAR4
SCHEMBL30454075 0.86 PTGER1 (0.47) MRGPRX4PTGER1
SCHEMBL30453291 0.86 C5AR1 (0.43) MRGPRX4DHODHNR4A2FFAR1PTGER1
SCHEMBL24257669 0.86 C5AR1 (0.43) MRGPRX4DHODHNR4A2FFAR1PTGER1
SCHEMBL24257585 0.86 PTGER1 (0.47) MRGPRX4PTGER1
Glycine SCHEMBL30546864 0.85 JAK2 (0.44) FFAR1FFAR4
SCHEMBL24257621 0.84 MCL1 (0.44) MCL1MRGPRX4DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230295110-A1 PHD INHIBITOR COMPOUNDS, COMPOSITIONS, AND METHODS OF USE AKEBIA THERAPEUTICS, INC. (US) 2023-09-21 US disclosed
US-20230295110-A1 PHD INHIBITOR COMPOUNDS, COMPOSITIONS, AND METHODS OF USE AKEBIA THERAPEUTICS, INC. (US) 2023-09-21 US disclosed
CN-116670131-A PHD inhibitor compounds, compositions, and methods of use 阿克比治疗有限公司 2023-08-29 CN disclosed
EP-4196466-A1 PHD INHIBITOR COMPOUNDS, COMPOSITIONS, AND METHODS OF USE Akebia Therapeutics Inc. (US) 2023-06-21 EP disclosed
WO-2022036188-A1 PHD INHIBITOR COMPOUNDS, COMPOSITIONS, AND METHODS OF USE AKEBIA THERAPEUTICS, INC. (US) 2022-02-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230295110-A1 PHD INHIBITOR COMPOUNDS, COMPOSITIONS, AND METHODS OF USE HIF1AN, EGLN3, PHF20 MCL1 2389/4885MRGPRX4 3994/4885DHODH 726/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.