SCHEMBL24257875

SCHEMBL24257875

N#Cc1ncc(Cl)c(C(F)F)c1Cl

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.44
CSNK1A1 P48729 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
CYP11B2 P19099 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2338301 0.76 KDM4E (0.53) KDM4EALDH1A1POLBCSNK1A1CLK4
SCHEMBL10387513 0.74
SCHEMBL30453863 0.72 LRRK2 (0.43) KDM4EALDH1A1
SCHEMBL24257841 0.72 LRRK2 (0.43) KDM4EALDH1A1
SCHEMBL18283690 0.71 POLB (0.48) KDM4EALDH1A1POLBCSNK1A1CLK4
SCHEMBL18283565 0.71 POLB (0.48) KDM4EALDH1A1POLBCSNK1A1CLK4
SCHEMBL27946108 0.68 KDM4E (0.41) KDM4EALDH1A1POLBCSNK1A1CLK4
SCHEMBL24257717 0.67 KDM4E (0.49) KDM4EALDH1A1POLBCSNK1A1CLK4
SCHEMBL30546876 0.67 KDM4E (0.49) KDM4EALDH1A1POLBCSNK1A1CLK4
SCHEMBL2331146 0.66 KDM4E (0.37) KDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230295110-A1 PHD INHIBITOR COMPOUNDS, COMPOSITIONS, AND METHODS OF USE AKEBIA THERAPEUTICS, INC. (US) 2023-09-21 US disclosed
US-20230295110-A1 PHD INHIBITOR COMPOUNDS, COMPOSITIONS, AND METHODS OF USE AKEBIA THERAPEUTICS, INC. (US) 2023-09-21 US disclosed
WO-2022036188-A1 PHD INHIBITOR COMPOUNDS, COMPOSITIONS, AND METHODS OF USE AKEBIA THERAPEUTICS, INC. (US) 2022-02-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230295110-A1 PHD INHIBITOR COMPOUNDS, COMPOSITIONS, AND METHODS OF USE HIF1AN, EGLN3, PHF20 KDM4E 175/4885ALDH1A1 1362/4885POLB 3169/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.