SCHEMBL24288652

SCHEMBL24288652

Cc1cccc2cc(-c3cccc4[nH]nc(N)c34)ccc12

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 20/20 0.66
KIT P10721 1/20 0.58
FLT3 P36888 1/20 0.58
LCK P06239 2/20 0.56
CSF1R P07333 2/20 0.56
FGFR1 P11362 2/20 0.56
PRKACA P17612 2/20 0.56
ROCK1 Q13464 2/20 0.56
PLK4 O00444 1/20 0.56
AURKA O14965 1/20 0.56
JAK2 O60674 1/20 0.56
CDK1 P06493 1/20 0.56
LYN P07948 1/20 0.56
SRC P12931 1/20 0.56
RPS6KB1 P23443 1/20 0.56
CDK2 P24941 1/20 0.56
MARK3 P27448 1/20 0.56
AKT1 P31749 1/20 0.56
AKT2 P31751 1/20 0.56
BLK P51451 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24288644 0.86 KDR (0.52) KDRKITFLT3CSF1RFGFR1
SCHEMBL24290092 0.83 KDR (0.53) KDRKITFLT3LCKCSF1R
SCHEMBL28871219 0.82 KDR (0.66) KDRKITFLT3LCKCSF1R
SCHEMBL29968063 0.82 KDR (0.66) KDRKITFLT3LCKCSF1R
SCHEMBL17034042 0.81 KDR (1.00) KDR
SCHEMBL29549949 0.81 KDR (1.00) KDR
SCHEMBL6013181 0.79 KDR (0.90) KDRKITFLT3LCKCSF1R
SCHEMBL419502 0.77 KDR (0.62) KDRKITFLT3LCKCSF1R
SCHEMBL29968270 0.77 KDR (0.62) KDRKITFLT3LCKCSF1R
SCHEMBL17034073 0.77 KDR (1.00) KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3112351-B1 NAPHTHYLAMIDE COMPOUND, PREPARATION METHOD AND USE THEREOF SHANGHAI INST MATERIA MEDICA CAS (CN) 2022-03-30 EP disclosed