SCHEMBL24317170

SCHEMBL24317170

CS(=O)(=O)c1ccc(Oc2cc(F)cc(C#N)c2)c2c1C(=O)C[C@H]2O

nearest known ligand 0.68

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 20/20 0.68
VEGFA P15692 4/20 0.65
CYP2C9 P11712 1/20 0.61
ARNT P27540 1/20 0.61
CYP2C19 P33261 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24317763 1.00 EPAS1 (0.68) EPAS1VEGFACYP2C9ARNTCYP2C19
SCHEMBL26812490 0.89 EPAS1 (0.67) EPAS1VEGFACYP2C9ARNTCYP2C19
SCHEMBL31404117 0.85 VEGFA (0.59) EPAS1VEGFA
SCHEMBL19870699 0.83 EPAS1 (0.67) EPAS1VEGFACYP2C9ARNTCYP2C19
SCHEMBL24317169 0.83 EPAS1 (0.70) EPAS1VEGFACYP2C9ARNTCYP2C19
SCHEMBL24317188 0.82 EPAS1 (0.66) EPAS1VEGFACYP2C9ARNTCYP2C19
SCHEMBL26812591 0.82 EPAS1 (0.72) EPAS1VEGFA
SCHEMBL16555409 0.81 EPAS1 (0.64) EPAS1VEGFA
SCHEMBL18036934 0.81 EPAS1 (1.00) EPAS1VEGFACYP2C9ARNTCYP2C19
SCHEMBL16560921 0.81 EPAS1 (1.00) EPAS1VEGFACYP2C9ARNTCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11827614-B2 Synthetic pathway to belzutifan and crystalline phases of synthetic intermediates MERCK SHARP & DOHME LLC (US) 2023-11-28 US disclosed
US-11827614-B2 Synthetic pathway to belzutifan and crystalline phases of synthetic intermediates MERCK SHARP & DOHME LLC (US) 2023-11-28 US disclosed
US-20220081407-A1 METHODS OF PREPARING SUBSTITUTED INDANES PELOTON THERAPEUTICS, INC. (US) 2022-03-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220081407-A1 METHODS OF PREPARING SUBSTITUTED INDANES HIF1AN, EGLN2, HIF1A EPAS1 25/4885VEGFA 1713/4885CYP2C9 1693/4885
US-11827614-B2 Synthetic pathway to belzutifan and crystalline phases of synthetic intermediates HIF1AN, HIF1A, EGLN2 EPAS1 18/4885VEGFA 115/4885CYP2C9 861/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.