SCHEMBL24327623

SCHEMBL24327623

CNc1ccc(Br)c2c1CCC2

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.33
HTR2A P28223 1/20 0.33
HTR2B P41595 1/20 0.33
NISCH Q9Y2I1 3/20 0.32
IL1RN P18510 1/20 0.31
ERAP2 Q6P179 1/20 0.31
ERAP1 Q9NZ08 1/20 0.31
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28753978 0.91 KDM4E (0.35) HTR2CHTR2AHTR2BIL1RNERAP2
SCHEMBL30509287 0.79 HTR2C (0.40) HTR2CHTR2AHTR2BIL1RNERAP2
SCHEMBL13249026 0.79 HTR2C (0.40) HTR2CHTR2AHTR2BIL1RNERAP2
SCHEMBL6674584 0.76 RXFP1 (0.51)
SCHEMBL13105773 0.74 NISCH (0.44) HTR2CHTR2AHTR2BNISCHKDM4E
SCHEMBL10463782 0.74 HTR2C (0.40) HTR2CHTR2AHTR2BIL1RNERAP2
SCHEMBL13249030 0.73 DRD4 (0.35) HTR2CNISCHIL1RNERAP2ERAP1
SCHEMBL21646755 0.72 USP2 (0.45) KDM4E
SCHEMBL2952459 0.72 RXFP1 (0.51)
SCHEMBL13585896 0.70 HTR2C (0.40) HTR2CHTR2AHTR2BIL1RNERAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022063106-A1 INDOLINE COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS BEIGENE, LTD. (KY) 2022-03-31 WO disclosed