SCHEMBL2432824

SCHEMBL2432824

COC(=O)[C@H]1CC[C@H](OC[C@@H]2CCCN2OCC(=O)Cc2ccc(NC(=O)c3cn(C)c4ccccc34)c(Cl)c2F)CC1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 13/20 0.56
ITGA4 P13612 13/20 0.56
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
KDM1A O60341 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GFER P55789 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7269962 1.00 ITGB1 (0.56) ITGB1ITGA4MEN1KMT2AKDM1A
SCHEMBL2432788 0.89 ITGB1 (0.71) ITGB1ITGA4MEN1KMT2AKDM1A
SCHEMBL2430237 0.89 ITGB1 (0.71) ITGB1ITGA4MEN1KMT2AKDM1A
SCHEMBL2432751 0.83 ITGB1 (0.80) ITGB1ITGA4
SCHEMBL2432856 0.83 ITGB1 (0.80) ITGB1ITGA4
SCHEMBL1170751 0.82 ITGB1 (0.70) ITGB1ITGA4MEN1KMT2AKDM1A
Water SCHEMBL2128631 0.82 ITGB1 (0.69) ITGB1ITGA4MEN1KMT2AKDM1A
Water SCHEMBL1170415 0.81 ITGB1 (0.61) ITGB1ITGA4MEN1KMT2AKDM1A
Bicarbonate SCHEMBL2438579 0.80 ITGB1 (0.60) ITGB1ITGA4MEN1KMT2AKDM1A
SCHEMBL2429857 0.79 ITGB1 (0.72) ITGB1ITGA4MEN1KMT2AKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346982-B1 VLA-4 INHIBITORS DAIICHI SEIYAKU CO (JP) 2011-09-14 EP disclosed